SCHEMBL17539693

SCHEMBL17539693

O=C(NCc1cccnc1)c1ccc(O)c(F)c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.64
ALDH1A1 P00352 3/20 0.61
L3MBTL1 Q9Y468 3/20 0.61
USP2 O75604 1/20 0.61
CA2 P00918 1/20 0.60
HTT P42858 2/20 0.60
LMNA P02545 2/20 0.60
MAPT P10636 1/20 0.60
CYP1A2 P05177 2/20 0.59
CYP3A4 P08684 2/20 0.59
TSHR P16473 2/20 0.59
BLM P54132 1/20 0.59
GAA P10253 1/20 0.58
CYP2C19 P33261 1/20 0.58
MAPK1 P28482 1/20 0.56
NAMPT P43490 1/20 0.56
VNN1 O95497 1/20 0.56
MMP13 P45452 2/20 0.55
CHRNB2 P17787 1/20 0.55
CHRNA7 P36544 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22972394 0.90 NPSR1 (0.64) NPSR1ALDH1A1L3MBTL1USP2CA2
SCHEMBL13504066 0.84 NPSR1 (0.60) NPSR1ALDH1A1L3MBTL1USP2CA2
SCHEMBL21246563 0.84 NPSR1 (0.62) NPSR1ALDH1A1L3MBTL1USP2CA2
SCHEMBL5783915 0.82 HTT (0.71) NPSR1ALDH1A1L3MBTL1CA2HTT
SCHEMBL3592277 0.82 POLB (0.63) NPSR1ALDH1A1L3MBTL1USP2CA2
SCHEMBL11628250 0.82 NPSR1 (0.67) NPSR1ALDH1A1L3MBTL1USP2HTT
SCHEMBL30491866 0.82 NPSR1 (0.67) NPSR1ALDH1A1L3MBTL1USP2HTT
SCHEMBL5257811 0.81 LMNA (0.72) NPSR1ALDH1A1CA2HTTLMNA
SCHEMBL19623369 0.79 ALDH1A1 (0.78) NPSR1ALDH1A1L3MBTL1USP2HTT
SCHEMBL7082686 0.79 TSHR (0.73) NPSR1ALDH1A1USP2CA2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2103613-B1 QUINOXALINE DERIVATIVE ASKA PHARM CO LTD (JP) 2016-02-17 EP disclosed