SCHEMBL17552175

SCHEMBL17552175

COc1ccc(C(=O)Nc2cccc3ccc(C)nc23)cc1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.62
TP53 P04637 2/20 0.62
KMT2A Q03164 5/20 0.62
NPC1 O15118 2/20 0.62
RAB9A P51151 1/20 0.62
F10 P00742 1/20 0.61
RXFP1 Q9HBX9 1/20 0.61
MAPT P10636 5/20 0.58
GAA P10253 1/20 0.58
ALDH1A1 P00352 2/20 0.58
MEN1 O00255 2/20 0.58
ALOX12 P18054 1/20 0.58
TSHR P16473 1/20 0.55
HSD17B10 Q99714 1/20 0.55
HDAC6 Q9UBN7 2/20 0.54
KDM4E B2RXH2 2/20 0.54
HDAC3 O15379 1/20 0.54
HDAC4 P56524 1/20 0.54
HDAC1 Q13547 1/20 0.54
HDAC7 Q8WUI4 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29911013 1.00 POLB (0.62) POLBTP53KMT2ANPC1RAB9A
SCHEMBL26798520 0.87 MAPT (0.64) POLBTP53KMT2ANPC1RAB9A
SCHEMBL17552186 0.86 KMT2A (0.74) POLBTP53KMT2ANPC1RAB9A
SCHEMBL17552230 0.86 MAPT (0.73) POLBTP53KMT2AMAPTGAA
SCHEMBL29831356 0.86 KMT2A (0.74) POLBTP53KMT2ANPC1RAB9A
SCHEMBL29911029 0.86 MAPT (0.73) POLBTP53KMT2AMAPTGAA
SCHEMBL29419544 0.86 MAPT (0.73) POLBTP53KMT2AMAPTGAA
SCHEMBL17540883 0.85 MAPT (0.58) POLBTP53KMT2ANPC1RAB9A
SCHEMBL17552254 0.85 MAPT (0.62) POLBTP53KMT2ANPC1RAB9A
SCHEMBL28154257 0.85 MAPT (0.76) POLBTP53KMT2ANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240016793-A1 QUINOLINES THAT MODULATE SERCA AND THEIR USE FOR TREATING DISEASE NEURODON CORPORATION 2024-01-18 US disclosed
US-11827626-B2 Quinolines that modulate SERCA and their use for treating disease NEURODON CORPORATION (US) 2023-11-28 US disclosed
EP-4037685-B1 QUINOLINE THAT MODULATE SERCA AND ITS USE FOR TREATING DISEASE NEURODON CORP (US) 2023-09-20 EP disclosed
US-20230285382-A1 QUINOLINES THAT MODULATE SERCA AND THEIR USE FOR TREATING DISEASE NEURODON CORPORATION 2023-09-14 US disclosed
CN-116744928-A Quinolines modulating SERCA and their use for treating diseases 神经元公司 2023-09-12 CN disclosed
US-11730729-B2 Quinolines that modulate SERCA and their use for treating disease NEURODON CORPORATION (US) 2023-08-22 US disclosed
US-20220016108-A1 QUINOLINES THAT MODULATE SERCA AND THEIR USE FOR TREATING DISEASE NEURODON CORPORATION 2022-01-20 US disclosed
US-20200347038-A1 QUINOLINES THAT MODULATE SERCA AND THEIR USE FOR TREATING DISEASE NEURODON CORPORATION 2020-11-05 US disclosed
US-20170281611-A1 QUINOLINES AND THEIR USE FOR TREATING ENDOPLASMIC RETICULUM STRESS-CAUSED DISEASES EIGER BIOPHARMACEUTICALS, INC. (US) 2017-10-05 US disclosed
WO-2016032569-A1 QUINOLINES AND THEIR USE FOR TREATING ENDOPLASMIC RETICULUM STRESS-CAUSED DISEASES CELLADON CORPORATION (US) 2016-03-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230285382-A1 QUINOLINES THAT MODULATE SERCA AND THEIR USE FOR TREATING DISEASE ATP2A1, ATP2A3, ATP2A2 POLB 3166/4885TP53 3732/4885KMT2A 4234/4885
US-20170281611-A1 QUINOLINES AND THEIR USE FOR TREATING ENDOPLASMIC RETICULUM STRESS-CAUSED DISEASES ATP2A1, ATP2A3, ATP2A2 POLB 2994/4885TP53 3254/4885KMT2A 4359/4885
US-11730729-B2 Quinolines that modulate SERCA and their use for treating disease ATP2A1, ATP2A3, ATP2A2 POLB 3166/4885TP53 3732/4885KMT2A 4234/4885
US-11827626-B2 Quinolines that modulate SERCA and their use for treating disease ATP2A1, ATP2A3, ATP2A2 POLB 3166/4885TP53 3732/4885KMT2A 4234/4885
US-20220016108-A1 QUINOLINES THAT MODULATE SERCA AND THEIR USE FOR TREATING DISEASE ATP2A1, ATP2A3, ATP2A2 POLB 3166/4885TP53 3732/4885KMT2A 4234/4885
US-20200347038-A1 QUINOLINES THAT MODULATE SERCA AND THEIR USE FOR TREATING DISEASE ATP2A1, ATP2A3, ATP2A2 POLB 3166/4885TP53 3732/4885KMT2A 4234/4885
US-20240016793-A1 QUINOLINES THAT MODULATE SERCA AND THEIR USE FOR TREATING DISEASE ATP2A1, ATP2A3, ATP2A2 POLB 3166/4885TP53 3732/4885KMT2A 4234/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.