SCHEMBL17554669

SCHEMBL17554669

O=C1CCc2cccc(Nc3ncc(F)c(CCc4ccc(Br)cc4F)n3)c2N1

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ULK1 O75385 4/20 0.38
PTK2 Q05397 7/20 0.37
NEK2 P51955 1/20 0.34
KDR P35968 3/20 0.34
MAOA P21397 2/20 0.32
MAOB P27338 2/20 0.32
KIF11 P52732 1/20 0.32
FLT4 P35916 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17554664 0.92 ULK1 (0.37) ULK1PTK2NEK2KDRFLT4
SCHEMBL670806 0.83 ULK1 (0.45) ULK1PTK2NEK2KDR
SCHEMBL15033827 0.81 ULK1 (0.56) ULK1PTK2KIF11
SCHEMBL669223 0.76 ULK1 (0.40) ULK1PTK2NEK2
SCHEMBL17554666 0.76 ULK1 (0.49) ULK1NEK2KDRMAOAMAOB
SCHEMBL15033846 0.75 ULK1 (0.56) ULK1PTK2KIF11
SCHEMBL15033850 0.75 PTK2B (0.52) ULK1PTK2KDR
SCHEMBL15033841 0.74 ULK1 (0.54) ULK1PTK2
SCHEMBL669259 0.74 ULK1 (0.43) ULK1PTK2NEK2KDRFLT4
SCHEMBL15033857 0.73 ULK1 (0.71) ULK1PTK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2606034-B1 PYRIMIDINE DERIVATIVE AS FAK INHIBITORS MERCK PATENT GMBH (DE) 2016-03-09 EP disclosed