SCHEMBL1755813

SCHEMBL1755813

COc1cc2c(cc1NO)Cc1c([nH]c3cc(Br)ccc13)C2(C)C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 13/20 0.44
GSK3B P49841 2/20 0.35
CCNB2 O95067 1/20 0.35
CDK1 P06493 1/20 0.35
CCNB1 P14635 1/20 0.35
CDK5 Q00535 1/20 0.35
CDK5R1 Q15078 1/20 0.35
CCNB3 Q8WWL7 1/20 0.35
CA1 P00915 2/20 0.34
CA2 P00918 2/20 0.34
CA4 P22748 2/20 0.34
CA6 P23280 2/20 0.34
TUBB4A P04350 1/20 0.33
TUBB P07437 1/20 0.33
TUBA3C P0DPH7 1/20 0.33
TUBA1B P68363 1/20 0.33
TUBA4A P68366 1/20 0.33
TUBB4B P68371 1/20 0.33
TUBB3 Q13509 1/20 0.33
TUBB2A Q13885 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL897744 0.86 ALK (0.50) ALKGSK3BCCNB2CDK1CCNB1
SCHEMBL16775676 0.85 ALK (0.47) ALKGSK3BCCNB2CDK1CCNB1
SCHEMBL27087539 0.84 ALK (0.48) ALKGSK3BCCNB2CDK1CCNB1
SCHEMBL897158 0.82 ALK (0.46) ALKGSK3BCCNB2CDK1CCNB1
SCHEMBL27087629 0.82 ALK (0.45) ALKGSK3BCCNB2CDK1CCNB1
SCHEMBL27087566 0.82 ALK (0.47) ALKGSK3BCCNB2CDK1CCNB1
SCHEMBL25446306 0.82 ALK (0.43) ALKGSK3BCCNB2CDK1CCNB1
SCHEMBL897277 0.80 ALK (0.45) ALKGSK3BCCNB2CDK1CCNB1
SCHEMBL896972 0.79 CDK4 (0.46) ALKGSK3BCCNB2CDK1CCNB1
SCHEMBL17448467 0.78 ALK (0.61) ALK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3613729-A1 TETRACYCLIC COMPOUNDS CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2020-02-26 EP disclosed
EP-3345903-B1 TETRACYCLIC COMPOUNDS CHUGAI PHARMACEUTICAL CO LTD (JP) 2019-10-09 EP disclosed
EP-3345903-A1 TETRACYCLIC COMPOUNDS Chugai Seiyaku Kabushiki Kaisha (JP) 2018-07-11 EP disclosed
EP-2975024-B1 TETRACYCLIC COMPOUNDS CHUGAI PHARMACEUTICAL CO LTD (JP) 2018-03-28 EP disclosed
EP-2975024-A1 TETRACYCLIC COMPOUNDS CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2016-01-20 EP disclosed
EP-2441753-A1 TETRACYCLIC COMPOUND Chugai Seiyaku Kabushiki Kaisha (JP) 2012-04-18 EP disclosed