SCHEMBL1755890

SCHEMBL1755890

CC(C)Oc1cc2c(cc1C1=CCN(C(=O)OC(C)(C)C)CC1)C(=O)c1c([nH]c3cc(N)ccc13)C2(C)C

nearest known ligand 0.49

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 18/20 0.49
PDK4 Q16654 1/20 0.47
CNR1 P21554 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7815079 0.92 ALK (0.51) ALKPDK4CNR1
SCHEMBL897569 0.90 ALK (0.60) ALK
SCHEMBL7816665 0.90 ALK (0.52) ALKPDK4CNR1
SCHEMBL7813080 0.86 ALK (0.54) ALKPDK4CNR1
SCHEMBL7806462 0.86 ALK (0.55) ALKPDK4CNR1
SCHEMBL7807827 0.83 ALK (0.60) ALK
SCHEMBL896882 0.82 ALK (0.62) ALK
SCHEMBL7806330 0.81 ALK (0.49) ALK
SCHEMBL1755858 0.80 ALK (0.48) ALK
SCHEMBL16776103 0.80 ALK (0.54) ALKPDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2441753-A1 TETRACYCLIC COMPOUND Chugai Seiyaku Kabushiki Kaisha (JP) 2012-04-18 EP disclosed
WO-2010143664-A1 TETRACYCLIC COMPOUND 中外製薬株式会社 (JP) 2010-12-16 WO disclosed