SCHEMBL1756033

SCHEMBL1756033

COC(=O)c1cccc(-c2cccc(N)c2O)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.51
CA9 Q16790 2/20 0.51
CA1 P00915 1/20 0.51
CA2 P00918 1/20 0.51
ERN1 O75460 5/20 0.50
PDK2 Q15119 1/20 0.49
ASH1L Q9NR48 1/20 0.48
LOXL2 Q9Y4K0 1/20 0.48
ALDH1A1 P00352 2/20 0.46
KDM4E B2RXH2 1/20 0.46
GLA P06280 1/20 0.46
GAA P10253 1/20 0.46
MAPT P10636 1/20 0.46
HPGD P15428 1/20 0.46
CASP1 P29466 1/20 0.46
CASP7 P55210 1/20 0.46
ATM Q13315 1/20 0.46
HSD17B10 Q99714 1/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL396896 0.88 CA12 (0.54) CA12CA9CA1CA2ERN1
SCHEMBL6736858 0.85 EGFR (0.56) CA12CA9CA1CA2ERN1
SCHEMBL28409132 0.82 ERN1 (0.50) CA12CA9CA1CA2ERN1
SCHEMBL29629597 0.81 KMO (0.53) CA12CA9CA1CA2ERN1
SCHEMBL407806 0.81 KMO (0.53) CA12CA9CA1CA2ERN1
SCHEMBL16749656 0.81 CA12 (0.58) CA12CA9CA1CA2ERN1
SCHEMBL6082886 0.80 EGFR (0.57) CA12CA9CA1CA2ERN1
Bromide SCHEMBL1706405 0.80 KMO (0.51) CA12CA9CA1CA2ERN1
Hydrochloric Acid SCHEMBL4861328 0.80 KMO (0.51) CA12CA9CA1CA2ERN1
SCHEMBL28755028 0.80 TSHR (0.60) CA12CA9CA1CA2ERN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2441457-A1 SALTS OF BICYCLO-SUBSTITUTED PYRAZOLON AZO DERIVATIVES, PREPARATION METHOD AND USE THEREOF Jiangsu Hengrui Medicine Co., Ltd. (CN) 2012-04-18 EP disclosed
EP-2236500-A1 BICYCLO-SUBSTITUTED PYRAZOLON AZO DERIVATIVES, PREPARATION PROCESS AND PHARMACEUTICAL USE THEREOF Jiangsu Hengrui Medicine Co., Ltd. (CN) 2010-10-06 EP disclosed