SCHEMBL17570698

SCHEMBL17570698

CNC(=O)NC(=O)CNC(=O)c1cc(OC)ccc1[N+](=O)[O-]

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.49
SMN1; SMN2 Q16637 5/20 0.43
AKR1B10 O60218 1/20 0.43
AKR1B1 P15121 1/20 0.43
AKR1C4 P17516 1/20 0.43
AKR1C3 P42330 1/20 0.43
AKR1C2 P52895 1/20 0.43
AKR1C1 Q04828 1/20 0.43
POLB P06746 1/20 0.43
MAPT P10636 4/20 0.42
NPC1 O15118 3/20 0.42
MAPK1 P28482 2/20 0.42
RAB9A P51151 2/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
CYP3A4 P08684 1/20 0.41
PSMB11 A5LHX3 1/20 0.41
PSMA7 O14818 1/20 0.41
PSMB1 P20618 1/20 0.41
PSMA1 P25786 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16840366 0.75 TAS1R3 (0.58) HPGDPOLBMAPTNPC1CYP3A4
SCHEMBL268414 0.74 TDP1 (0.62) HPGDSMN1; SMN2AKR1B10AKR1B1AKR1C4
SCHEMBL14373412 0.73 HPGD (0.45) HPGDSMN1; SMN2POLBNPC1MEN1
SCHEMBL12326834 0.72 ALDH1A1 (0.53) HPGDSMN1; SMN2AKR1B10AKR1B1AKR1C4
SCHEMBL269614 0.72 AKR1C3 (0.63) HPGDSMN1; SMN2AKR1B10AKR1B1AKR1C4
SCHEMBL30580504 0.72 AKR1C3 (0.63) HPGDSMN1; SMN2AKR1B10AKR1B1AKR1C4
SCHEMBL4273530 0.72 SMN1; SMN2 (0.52) HPGDSMN1; SMN2AKR1B10AKR1B1AKR1C4
SCHEMBL404510 0.71 MAPT (0.51) HPGDSMN1; SMN2AKR1B10AKR1B1AKR1C4
SCHEMBL4946199 0.71 AKR1C3 (0.51) HPGDSMN1; SMN2AKR1B10AKR1B1AKR1C4
Potassium Ion SCHEMBL15876122 0.71 AKR1C3 (0.51) HPGDSMN1; SMN2AKR1B10AKR1B1AKR1C4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1976849-B1 COMPOUNDS FOR THE TREATMENT OF INFLAMMATORY DISORDERS MERCK SHARP & DOHME (US) 2016-03-09 EP disclosed