SCHEMBL1758672

SCHEMBL1758672

O=C(Cc1csc(CCCCC23CC4CC(CC(C4)C2)C3)n1)NO

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 16/20 0.41
HDAC6 Q9UBN7 16/20 0.41
PDE5A O76074 3/20 0.40
PDE1A P54750 1/20 0.40
PDE1B Q01064 1/20 0.40
PDE1C Q14123 1/20 0.40
HDAC3 O15379 3/20 0.38
HDAC4 P56524 3/20 0.38
HDAC7 Q8WUI4 3/20 0.38
HDAC2 Q92769 3/20 0.38
HDAC10 Q969S8 3/20 0.38
HDAC11 Q96DB2 3/20 0.38
HDAC8 Q9BY41 3/20 0.38
HDAC9 Q9UKV0 3/20 0.38
HDAC5 Q9UQL6 3/20 0.38
KDM4E B2RXH2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6878807 0.88 HDAC1 (0.36) HDAC1HDAC6PDE5APDE1APDE1B
SCHEMBL1758740 0.78 PDE5A (0.37) HDAC1HDAC6PDE5APDE1APDE1B
SCHEMBL1758679 0.76 PDE5A (0.41) HDAC6PDE5APDE1APDE1BPDE1C
SCHEMBL1758713 0.74 PDE5A (0.54) PDE5APDE1APDE1BPDE1CKDM4E
SCHEMBL1758576 0.74 HDAC1 (0.51) HDAC1HDAC6HDAC3HDAC4HDAC7
SCHEMBL1758697 0.74 PDE5A (0.40) HDAC1HDAC6PDE5APDE1APDE1B
SCHEMBL15522909 0.73 HDAC1 (0.67) HDAC1HDAC6PDE5APDE1APDE1B
SCHEMBL6881726 0.72 HPGD (0.41)
SCHEMBL1758588 0.71 MEN1 (0.34)
SCHEMBL1759205 0.71 CNR2 (0.62) PDE5APDE1APDE1BPDE1CKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011058582-A1 HISTONE DEACETYLASE INHIBITORS FOR THE TREATMENT OF FUNGAL INFECTIONS ORCHID RESEARCH LABORATORIES LTD. (IN) 2011-05-19 WO claimed
WO-2011058582-A1 HISTONE DEACETYLASE INHIBITORS FOR THE TREATMENT OF FUNGAL INFECTIONS ORCHID RESEARCH LABORATORIES LTD. (IN) 2011-05-19 WO disclosed