SCHEMBL17591561

SCHEMBL17591561

OCCOc1ccncn1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.39
RECQL P46063 1/20 0.39
CYP2D6 P10635 2/20 0.39
HSP90AA1 P07900 1/20 0.37
P2RX7 Q99572 1/20 0.36
THRB P10828 1/20 0.35
KMT2A Q03164 1/20 0.35
LOX P28300 1/20 0.34
AOC3 Q16853 1/20 0.34
PIK3CD O00329 1/20 0.34
PIK3CA P42336 1/20 0.34
PIK3CB P42338 1/20 0.34
PI4KA P42356 1/20 0.34
PIK3CG P48736 1/20 0.34
PI4KB Q9UBF8 1/20 0.34
SORD Q00796 1/20 0.33
CYP3A4 P08684 1/20 0.32
NR1I2 O75469 1/20 0.32
GCK P35557 1/20 0.32
IDO1 P14902 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27890075 0.88 LOX (0.39) CYP2D6HSP90AA1P2RX7LOXAOC3
SCHEMBL22110815 0.83 HSP90AA1 (0.37) CYP2D6HSP90AA1P2RX7RXRAGRIN1
SCHEMBL8566274 0.79 HSP90AA1 (0.37) CYP2D6HSP90AA1P2RX7RXRAGRIN1
SCHEMBL19732852 0.79 HSP90AA1 (0.41) CYP2D6HSP90AA1P2RX7
SCHEMBL27906749 0.78 IRAK4 (0.32) CYP2D6HSP90AA1P2RX7THRBRXRA
SCHEMBL6638944 0.78 CYP2D6 (0.57) ALDH1A1CYP2D6CYP3A4
SCHEMBL27890125 0.76 CYP19A1 (0.36) ALDH1A1CYP2D6HSP90AA1P2RX7IDO1
SCHEMBL27890078 0.76 P2RX7 (0.35) ALDH1A1CYP2D6HSP90AA1P2RX7IDO1
SCHEMBL28803714 0.74 CYP2D6 (0.36) CYP2D6HSP90AA1P2RX7CYP3A4RXRA
SCHEMBL5883850 0.74

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102924446-A PIM kinase inhibitor, preparation method thereof, and application thereof in pharmacy SHANGHAI JIKAI MEDICAL TECHNOLOGY CO LTD 2013-02-13 CN claimed
EP-2804854-B1 SUBSTITUTED TRIAZOLES AND THEIR USE FOR TREATMENT AND/OR PREVENTION OF NEUROLOGICAL AND PSYCHIATRIC DISORDERS BOEHRINGER INGELHEIM INT (DE) 2016-03-16 EP disclosed
CN-102924446-A PIM kinase inhibitor, preparation method thereof, and application thereof in pharmacy SHANGHAI JIKAI MEDICAL TECHNOLOGY CO LTD 2013-02-13 CN disclosed