SCHEMBL1759218

SCHEMBL1759218

COC(=O)NC(CO)Cc1cn(Cc2ccccc2)nn1

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 7/20 0.48
HDAC1 Q13547 1/20 0.47
HSP90AB1 P08238 2/20 0.46
ALDH1A1 P00352 1/20 0.46
LMNA P02545 1/20 0.46
OPRM1 P35372 1/20 0.44
OPRD1 P41143 1/20 0.44
OPRK1 P41145 1/20 0.44
HRH4 Q9H3N8 1/20 0.44
MME P08473 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1838394 0.87 CYP19A1 (0.51) CYP19A1HDAC1HSP90AB1ALDH1A1LMNA
SCHEMBL305197 0.85 CYP19A1 (0.49) CYP19A1HDAC1HSP90AB1ALDH1A1LMNA
SCHEMBL14479459 0.81 CYP19A1 (0.48) CYP19A1HDAC1HSP90AB1ALDH1A1LMNA
SCHEMBL18183893 0.81 CYP19A1 (0.48) CYP19A1HDAC1HSP90AB1ALDH1A1LMNA
SCHEMBL19701642 0.79 CYP19A1 (0.43) CYP19A1HDAC1HSP90AB1ALDH1A1LMNA
SCHEMBL3097402 0.76 CYP19A1 (0.57) CYP19A1HDAC1HSP90AB1ALDH1A1LMNA
SCHEMBL29255128 0.76 ALDH1A1 (0.50) CYP19A1HDAC1ALDH1A1LMNAMME
SCHEMBL24666587 0.75 CYP19A1 (0.57) CYP19A1HDAC1HSP90AB1ALDH1A1LMNA
SCHEMBL3331695 0.75 ACE (0.56) MME
SCHEMBL304588 0.75 ACE (0.56) MME

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2513091-A1 HEPATITIS C VIRUS INHIBITORS Bristol-Myers Squibb Company (US) 2012-10-24 EP disclosed
EP-2499115-A1 HEPATITIS C VIRUS INHIBITORS Bristol-Myers Squibb Company (US) 2012-09-19 EP disclosed
EP-2499127-A1 HEPATITIS C VIRUS INHIBITORS Bristol-Myers Squibb Company (US) 2012-09-19 EP disclosed
WO-2011075439-A1 HEPATITIS C VIRUS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2011-06-23 WO disclosed
WO-2011059850-A1 HEPATITIS C VIRUS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2011-05-19 WO disclosed
WO-2011059887-A1 HEPATITIS C VIRUS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2011-05-19 WO disclosed