SCHEMBL17595043

SCHEMBL17595043

CCc1cc(C(=O)OC(=O)C(F)(F)F)c(=O)[nH]c1-c1ccc(N2CC3OCCN(Cc4ccccc4)C3C2)cc1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 2/20 0.34
PDE3A Q14432 2/20 0.34
CHRM4 P08173 4/20 0.32
CHRM2 P08172 2/20 0.31
CHRM1 P11229 2/20 0.31
CHRM5 P08912 1/20 0.31
CHRM3 P20309 1/20 0.31
TACR1 P25103 3/20 0.31
TACR2 P21452 1/20 0.31
TACR3 P29371 1/20 0.31
ALDH1A1 P00352 3/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
GAA P10253 2/20 0.31
RXFP1 Q9HBX9 1/20 0.30
KDM4E B2RXH2 1/20 0.30
POLB P06746 1/20 0.30
MAPT P10636 1/20 0.30
ALOX15 P16050 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL14741065 0.90 L3MBTL1 (0.34) PDE3BPDE3ACHRM2CHRM1ALDH1A1
SCHEMBL14758823 0.89 PDE3B (0.34) PDE3BPDE3AALDH1A1SMN1; SMN2MEN1
SCHEMBL14745349 0.88 ADK (0.38) PDE3BPDE3A
SCHEMBL14744863 0.77 HRH3 (0.41) MAPT
Trifluoroacetic Acid SCHEMBL14745348 0.77 ADK (0.40)
SCHEMBL14745225 0.77 PRKD3 (0.44) PDE3BPDE3AMAPT
SCHEMBL16568097 0.77 KCNH2 (0.33) ALDH1A1KDM4EMAPT
SCHEMBL14745525 0.76 PDE3B (0.34) PDE3BPDE3ACHRM4
SCHEMBL14745785 0.76 CHRM4 (0.36) PDE3BPDE3ACHRM4CHRM2CHRM1
SCHEMBL14745048 0.75 CHRM4 (0.35) PDE3BPDE3ACHRM4CHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016039936-A2 MONOCYCLIC SUBSTITUTED 2-PYRIDINONE ANTIBACTERIAL COMPOUNDS PTC THERAPEUTICS, INC. (US) 2016-03-17 WO claimed