SCHEMBL17595084

SCHEMBL17595084

CCc1c(-c2ccc(N3CCOCC3)cn2)[nH]c(=O)c(C(=O)O)c1O.CCc1cc(C(=O)O)c(=O)[nH]c1-c1ccc(N2CCC2)cc1.CCc1cc(C(=O)O)c(=O)[nH]c1-c1ccc(N2CCOCC2)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 9/20 0.36
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 2/20 0.35
POLB P06746 2/20 0.35
TDP1 Q9NUW8 2/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
MAPT P10636 1/20 0.35
DNMT1 P26358 1/20 0.35
APEX1 P27695 1/20 0.35
RECQL P46063 1/20 0.35
CACNA1B Q00975 1/20 0.35
APBA1 Q02410 1/20 0.35
CTDSP1 Q9GZU7 1/20 0.35
PARP2 Q9UGN5 3/20 0.34
MAP3K11 Q16584 1/20 0.33
ALK Q9UM73 1/20 0.33
LMNA P02545 1/20 0.33
MAP4K1 Q92918 1/20 0.32
TNKS O95271 1/20 0.32
PARP6 Q2NL67 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14740870 0.88 PARP1 (0.39) PARP1KDM4EALDH1A1POLBTDP1
SCHEMBL17594868 0.85 KIF11 (0.38) PARP1ALDH1A1L3MBTL1PARP2LMNA
SCHEMBL17594969 0.84 KIF11 (0.39) PARP1ALDH1A1PARP2LMNAMEN1
SCHEMBL17595085 0.84 PARP1 (0.32) PARP1PARP2
SCHEMBL14740829 0.81 SLC16A3 (0.45) PARP1KDM4EALDH1A1POLBTDP1
SCHEMBL14745174 0.79 KCNH2 (0.40) PARP1ALDH1A1POLBMAPTPARP2
SCHEMBL14741099 0.79 PARP1 (0.41) PARP1KDM4EALDH1A1L3MBTL1MAPT
SCHEMBL14745530 0.78 KDM4E (0.39) PARP1KDM4EALDH1A1PARP2TNKS
SCHEMBL14747044 0.77 KIF11 (0.41) PARP1ALDH1A1POLBL3MBTL1MAPT
SCHEMBL14745092 0.77 PARP1 (0.43) PARP1ALDH1A1L3MBTL1MAPTPARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016039936-A2 MONOCYCLIC SUBSTITUTED 2-PYRIDINONE ANTIBACTERIAL COMPOUNDS PTC THERAPEUTICS, INC. (US) 2016-03-17 WO claimed