SCHEMBL17595085

SCHEMBL17595085

CCc1cc(C(=O)OC(=O)c2cc(CC)c(-c3ccc(N4CCC4)cc3)n(OC(=O)c3c(O)c(CC)c(-c4ccc(N5CCOCC5)cn4)[nH]c3=O)c2=O)c(=O)[nH]c1-c1ccc(N2CCOCC2)cc1

nearest known ligand 0.32

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.32
PARP2 Q9UGN5 1/20 0.32
SIRT2 Q8IXJ6 1/20 0.31
SIRT1 Q96EB6 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17595084 0.84 PARP1 (0.36) PARP1PARP2
SCHEMBL17594871 0.79 ALDH1A1 (0.39) PARP1PARP2SIRT2SIRT1
SCHEMBL17594971 0.78 LMNA (0.39) PARP1PARP2SIRT2SIRT1
SCHEMBL14740870 0.74 PARP1 (0.39) PARP1PARP2
SCHEMBL17594868 0.69 KIF11 (0.38) PARP1PARP2SIRT2SIRT1
SCHEMBL14745803 0.68 DCTPP1 (0.40) PARP1PARP2SIRT2SIRT1
SCHEMBL17594969 0.68 KIF11 (0.39) PARP1PARP2SIRT2SIRT1
SCHEMBL17595142 0.68 ABCB1 (0.39)
SCHEMBL14740829 0.67 SLC16A3 (0.45) PARP1PARP2SIRT2SIRT1
SCHEMBL17595256 0.67 PDE3B (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016039936-A2 MONOCYCLIC SUBSTITUTED 2-PYRIDINONE ANTIBACTERIAL COMPOUNDS PTC THERAPEUTICS, INC. (US) 2016-03-17 WO claimed