SCHEMBL17599487

SCHEMBL17599487

O=C(O)[C@@H]1CCN(c2ccc([N+](=O)[O-])c3ccccc23)C1

nearest known ligand 0.59

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CTSB P07858 4/20 0.59
AR P10275 4/20 0.59
NOTUM Q6P988 6/20 0.56
TDP1 Q9NUW8 1/20 0.54
KEAP1 Q14145 3/20 0.49
NFE2L2 Q16236 1/20 0.49
KMT2A Q03164 1/20 0.47
ALDH1A1 P00352 1/20 0.47
LMNA P02545 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17599443 1.00 CTSB (0.59) CTSBARNOTUMTDP1KEAP1
SCHEMBL5240888 0.92 CTSB (0.66) CTSBARTDP1KMT2AALDH1A1
SCHEMBL2559524 0.84 NOTUM (0.65) NOTUMTDP1KMT2AALDH1A1LMNA
SCHEMBL17599441 0.79 NOTUM (0.61) NOTUMKEAP1NFE2L2
SCHEMBL17612866 0.79 NOTUM (0.61) NOTUMKEAP1NFE2L2
SCHEMBL24811432 0.79 NOTUM (0.61) NOTUMKEAP1NFE2L2
SCHEMBL4879663 0.78 CTSB (0.74) CTSBARTDP1KMT2AALDH1A1
SCHEMBL2558464 0.78 NOTUM (0.56) NOTUMTDP1KMT2AALDH1A1
SCHEMBL2553837 0.78 NOTUM (0.56) NOTUMTDP1KMT2AALDH1A1LMNA
SCHEMBL2559422 0.77 ALDH1A1 (0.69) CTSBNOTUMTDP1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2997966-A1 Naphthyl Sulfonamide Pyrrolidine Derivatives as KEAP-1 Modulators for the Treatment of Diabetes, Obesity, Dyslipidemia and Related Disorders SANOFI (FR) 2016-03-23 EP disclosed