SCHEMBL176007

SCHEMBL176007

Nc1ccccc1-c1ncc(C(=O)c2ccccc2)s1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 10/20 0.66
RAB9A P51151 10/20 0.66
MAPT P10636 8/20 0.66
ALDH1A1 P00352 7/20 0.66
SMN1; SMN2 Q16637 6/20 0.66
NFKB1 P19838 2/20 0.58
NFKB2 Q00653 2/20 0.58
RELA Q04206 2/20 0.58
PPARG P37231 1/20 0.58
NCOA2 Q15596 1/20 0.58
NCOA1 Q15788 1/20 0.58
NCOA3 Q9Y6Q9 1/20 0.58
CYP1A2 P05177 3/20 0.55
CYP3A4 P08684 2/20 0.55
CYP2C9 P11712 2/20 0.55
CYP2C19 P33261 2/20 0.55
MAPK13 O15264 1/20 0.50
MAPK12 P53778 1/20 0.50
MAPK11 Q15759 1/20 0.50
MAPK14 Q16539 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12788381 0.80 NPC1 (1.00) NPC1RAB9AMAPTALDH1A1SMN1; SMN2
SCHEMBL6319469 0.78 NPC1 (0.63) NPC1RAB9AMAPTALDH1A1SMN1; SMN2
SCHEMBL6481114 0.74 NPC1 (0.88) NPC1RAB9AMAPTALDH1A1SMN1; SMN2
SCHEMBL1207792 0.73 PTPN1 (0.51) NPC1RAB9AMAPTALDH1A1SMN1; SMN2
SCHEMBL12745815 0.72 NPC1 (0.60) NPC1RAB9AMAPTALDH1A1SMN1; SMN2
SCHEMBL4283915 0.71 HPGD (0.55) NPC1RAB9AMAPTALDH1A1SMN1; SMN2
SCHEMBL1207018 0.71 ALDH1A1 (0.47) NPC1RAB9AMAPTALDH1A1SMN1; SMN2
SCHEMBL27768717 0.71 NPC1 (0.83) NPC1RAB9AMAPTALDH1A1SMN1; SMN2
SCHEMBL6482978 0.71 NPC1 (0.80) NPC1RAB9AMAPTALDH1A1SMN1; SMN2
SCHEMBL892320 0.70 ALDH1A1 (0.44) NPC1RAB9AMAPTALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012028100-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-08 WO disclosed