SCHEMBL1760842

SCHEMBL1760842

COc1ccnc2sc(NC(=O)N3CCC(N)C3)nc12

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 14/20 0.50
ADORA1 P30542 12/20 0.50
ADORA2B P29275 2/20 0.44
ADORA3 P0DMS8 1/20 0.44
ALDH1A1 P00352 2/20 0.44
MAPT P10636 1/20 0.44
TSHR P16473 1/20 0.44
HSD17B10 Q99714 1/20 0.44
PIM2 Q9P1W9 1/20 0.42
HDAC1 Q13547 1/20 0.41
HDAC2 Q92769 1/20 0.41
KDM4E B2RXH2 1/20 0.40
HPGD P15428 1/20 0.40
DYRK1A Q13627 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12592956 1.00 ADORA2A (0.50) ADORA2AADORA1ADORA2BADORA3ALDH1A1
SCHEMBL12592880 0.83 ADORA2A (0.42) ADORA2AADORA1ADORA2BADORA3ALDH1A1
SCHEMBL1760963 0.83 ADORA2A (0.42) ADORA2AADORA1ADORA2BADORA3ALDH1A1
SCHEMBL1760877 0.83 ADORA2A (0.42) ADORA2AADORA1ADORA2BADORA3ALDH1A1
SCHEMBL12592953 0.82 CFTR (0.50) ADORA2AADORA1ADORA2BADORA3HDAC1
SCHEMBL1760993 0.82 CFTR (0.50) ADORA2AADORA1ADORA2BADORA3HDAC1
SCHEMBL1760991 0.76 ADORA2A (0.46) ADORA2AADORA1ADORA2BADORA3ALDH1A1
SCHEMBL1761044 0.75 ADORA2A (0.40) ADORA2AADORA1ADORA2B
SCHEMBL12592960 0.75 ADORA2A (0.40) ADORA2AADORA1ADORA2B
SCHEMBL22063329 0.74 ADORA2A (0.42) ADORA2AADORA1ALDH1A1MAPTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7947692-B2 Substituted thiazolo[5,4-d]pyrimidine urea derivatives HOFFMANN-LA ROCHE INC. (US) 2011-05-24 US disclosed