SCHEMBL1761044

SCHEMBL1761044

COc1ccnc2sc(NC(=O)N3CCC(NCc4ccc(F)c(C(F)(F)F)c4)C3)nc12

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 15/20 0.40
ADORA1 P30542 13/20 0.40
ADORA2B P29275 6/20 0.40
PIK3CD O00329 1/20 0.38
PIK3CA P42336 1/20 0.38
TEAD1 P28347 2/20 0.37
SCD O00767 1/20 0.37
ENPP2 Q13822 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12592960 1.00 ADORA2A (0.40) ADORA2AADORA1ADORA2BPIK3CDPIK3CA
SCHEMBL2929522 0.89 ADORA2B (0.37) ADORA2AADORA1ADORA2BSCD
SCHEMBL1760967 0.88 PIK3CD (0.42) ADORA2AADORA1ADORA2BPIK3CDPIK3CA
SCHEMBL12592897 0.88 PIK3CD (0.42) ADORA2AADORA1ADORA2BPIK3CDPIK3CA
SCHEMBL1761043 0.84 PIK3CD (0.40) ADORA2AADORA1ADORA2BPIK3CDPIK3CA
SCHEMBL2931938 0.77 PIK3CD (0.37) ADORA2AADORA1ADORA2BPIK3CDPIK3CA
SCHEMBL3047619 0.76 RIPK1 (0.37) ADORA2AADORA1ADORA2BPIK3CDPIK3CA
SCHEMBL1760993 0.76 CFTR (0.50) ADORA2AADORA1ADORA2B
SCHEMBL12592953 0.76 CFTR (0.50) ADORA2AADORA1ADORA2B
SCHEMBL1760842 0.75 ADORA2A (0.50) ADORA2AADORA1ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7947692-B2 Substituted thiazolo[5,4-d]pyrimidine urea derivatives HOFFMANN-LA ROCHE INC. (US) 2011-05-24 US disclosed