SCHEMBL17609153

SCHEMBL17609153

COc1ccc(N(C)c2ccc(Oc3ccccn3)cc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.45
HTT P42858 1/20 0.45
RAB9A P51151 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
RXFP1 Q9HBX9 1/20 0.45
CASP1 P29466 1/20 0.43
CASP14 P31944 1/20 0.43
CASP3 P42574 1/20 0.43
CASP2 P42575 1/20 0.43
CASP4 P49662 1/20 0.43
CASP5 P51878 1/20 0.43
CASP7 P55210 1/20 0.43
CASP9 P55211 1/20 0.43
CASP6 P55212 1/20 0.43
CASP8 Q14790 1/20 0.43
CASP12 Q6UXS9 1/20 0.43
CASP10 Q92851 1/20 0.43
LTA4H P09960 2/20 0.43
EGFR P00533 3/20 0.43
PDGFRB P09619 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17602080 0.90 LTA4H (0.44) LTA4HEGFRPTGS2CSF1RMEN1
SCHEMBL17602116 0.89 LTA4H (0.43) NPC1HTTRAB9ALTA4HPTGS2
SCHEMBL18984681 0.88 RAB9A (0.54) NPC1HTTRAB9ANPSR1RXFP1
SCHEMBL17609125 0.88 MEN1 (0.45) NPC1HTTRAB9ACASP3LTA4H
SCHEMBL17602309 0.86 MAPK1 (0.48) HTTRAB9ALTA4HPTGS2PGR
SCHEMBL17609138 0.84 KDM4C (0.50) LTA4HPTGS2LMNAKDM4EALDH1A1
SCHEMBL17602142 0.84 KDM4C (0.47) LTA4HPTGS2CSF1RKDM4EDRD1
SCHEMBL17602209 0.84 KDM4C (0.44) NPC1RAB9ALTA4HEGFRPDGFRB
SCHEMBL17602210 0.84 KAT2B (0.45) NPC1RAB9ALTA4HPTGS2LMNA
SCHEMBL17602207 0.84 RAB9A (0.48) NPC1HTTRAB9ANPSR1LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3193601-A1 HISTONE DEMETHYLASE INHIBITORS Celgene Quanticel Research, Inc. (US) 2017-07-26 EP disclosed
WO-2016044429-A1 HISTONE DEMETHYLASE INHIBITORS Quanticel Pharmaceuticals, Inc. (US) 2016-03-24 WO disclosed