SCHEMBL176991

SCHEMBL176991

CN[C@@H](C)C(N)[C@@H](C(=O)N1CCC[C@H]1C(=O)Nc1cc2c(Nc3ccc4[nH]ncc4c3)ncnc2cc1OC)C(C)(C)C

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EGFR P00533 10/20 0.56
CYP3A4 P08684 7/20 0.54
CYP2C9 P11712 2/20 0.54
CYP2C19 P33261 1/20 0.54
XIAP P98170 1/20 0.54
RET P07949 3/20 0.49
ERBB2 P04626 4/20 0.44
KDR P35968 3/20 0.42
EP300 Q09472 1/20 0.42
ERBB4 Q15303 2/20 0.41
RAF1 P04049 2/20 0.40
FGFR2 P21802 2/20 0.40
FLT4 P35916 2/20 0.40
TEK Q02763 2/20 0.40
ABL1 P00519 1/20 0.40
LCK P06239 1/20 0.40
SRC P12931 1/20 0.40
FLT1 P17948 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL160911 0.87 CYP3A4 (0.72) EGFRCYP3A4CYP2C9CYP2C19XIAP
SCHEMBL160910 0.87 CYP3A4 (0.72) EGFRCYP3A4CYP2C9CYP2C19XIAP
SCHEMBL168498 0.86 CYP3A4 (0.58) EGFRCYP3A4CYP2C9CYP2C19XIAP
Hydrochloric Acid SCHEMBL176332 0.83 CYP3A4 (0.55) EGFRCYP3A4CYP2C9CYP2C19XIAP
SCHEMBL178188 0.83 CYP3A4 (0.58) EGFRCYP3A4CYP2C9CYP2C19XIAP
SCHEMBL176198 0.83 CYP3A4 (0.54) EGFRCYP3A4CYP2C9CYP2C19XIAP
Hydrochloric Acid SCHEMBL176203 0.83 CYP3A4 (0.56) EGFRCYP3A4CYP2C9CYP2C19XIAP
Hydrochloric Acid SCHEMBL176337 0.81 CYP3A4 (0.54) EGFRCYP3A4CYP2C9CYP2C19XIAP
SCHEMBL15050653 0.81 CYP3A4 (0.58) EGFRCYP3A4CYP2C9CYP2C19XIAP
SCHEMBL176377 0.81 EGFR (0.61) EGFRCYP3A4ERBB2ERBB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2611797-A2 QUINOLINE OR QUINAZOLINE DERIVATIVES WITH APOPTOSIS INDUCING ACTIVITY ON CELLS Hanmi Science Co., Ltd. (KR) 2013-07-10 EP disclosed
WO-2012030160-A2 QUINOLINE OR QUINAZOLINE DERIVATIVES WITH APOPTOSIS INDUCING ACTIVITY ON CELLS HANMI HOLDINGS CO., LTD. (KR) 2012-03-08 WO disclosed