SCHEMBL17620892

SCHEMBL17620892

COc1cccc(OC)c1CNC(=N)Nc1ccc(-c2ccc(F)cc2)cn1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.47
ABCB1 P08183 4/20 0.43
ABCC1 P33527 3/20 0.43
MAPK1 P28482 6/20 0.41
PSEN1 P49768 2/20 0.40
PSEN2 P49810 2/20 0.40
APH1B Q8WW43 2/20 0.40
NCSTN Q92542 2/20 0.40
APH1A Q96BI3 2/20 0.40
PSENEN Q9NZ42 2/20 0.40
WNT3A P56704 2/20 0.39
KDR P35968 1/20 0.38
TEK Q02763 1/20 0.38
FYN P06241 1/20 0.38
PDGFRB P09619 1/20 0.38
PDGFRA P16234 1/20 0.38
GPR55 Q9Y2T6 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acetic Acid SCHEMBL2781275 0.95 ROCK2 (0.48) ROCK2ABCB1ABCC1MAPK1WNT3A
SCHEMBL2779993 0.92 ROCK2 (0.47) ROCK2ABCB1ABCC1WNT3A
Acetic Acid SCHEMBL2781387 0.88 ROCK2 (0.49) ROCK2ABCB1ABCC1WNT3A
SCHEMBL17620898 0.88 KMT2A (0.48) ROCK2ABCB1ABCC1MAPK1
SCHEMBL2782249 0.84 MAPK1 (0.43) ROCK2MAPK1
SCHEMBL2780845 0.83 KMT2A (0.51) ROCK2MAPK1
Acetic Acid SCHEMBL2781206 0.83 HTT (0.49) ROCK2ABCB1ABCC1MAPK1
SCHEMBL2784131 0.82 ROCK2 (0.42) ROCK2MAPK1
SCHEMBL2783259 0.82 SCN9A (0.44) ROCK2
SCHEMBL2781082 0.81 MAPK1 (0.51) MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9296697-B2 Hetaryl-substituted guanidine compounds and use thereof as binding partners for 5-HT5-receptors ABBOTT LABORATORIES (US) 2016-03-29 US claimed