SCHEMBL17620893

SCHEMBL17620893

COc1cccc(OC)c1CNC(N)=Nc1ccc(-c2ccc(F)cc2)cn1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
FYN P06241 5/20 0.42
ROCK2 O75116 2/20 0.41
KIT P10721 2/20 0.41
MAP3K11 Q16584 2/20 0.38
PDGFRB P09619 1/20 0.38
PDGFRA P16234 1/20 0.38
MAPK1 P28482 2/20 0.36
POLB P06746 1/20 0.36
KMT2A Q03164 1/20 0.36
PRMT5 O14744 1/20 0.36
WDR77 Q9BQA1 1/20 0.36
LMNA P02545 1/20 0.36
HTT P42858 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
SMO Q99835 1/20 0.36
ROCK1 Q13464 1/20 0.35
DHPS P49366 1/20 0.35
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2779998 0.92 ROCK2 (0.42) FYNROCK2KITPDGFRBPDGFRA
SCHEMBL2782255 0.85 PLAU (0.41) FYNROCK2KITMAP3K11MAPK1
SCHEMBL2780849 0.84 ADRA2A (0.50) ROCK2MAPK1POLBKMT2ALMNA
SCHEMBL2781278 0.83 ROCK2 (0.42) FYNROCK2PDGFRBPDGFRAMAPK1
SCHEMBL2784134 0.83 ROCK2 (0.36) ROCK2MAPK1NPSR1DHPSALDH1A1
SCHEMBL2783265 0.82 SCN9A (0.40) ROCK2MAPK1POLBKMT2ALMNA
SCHEMBL2781085 0.81 MAPK1 (0.46) ROCK2MAPK1ROCK1ALDH1A1
SCHEMBL2781942 0.81 HTT (0.52) ROCK2POLBKMT2ALMNAHTT
SCHEMBL2782470 0.81 MAPK1 (0.43) ROCK2MAPK1ROCK1ALDH1A1
SCHEMBL2379939 0.81 PRMT5 (0.44) FYNROCK2KITMAPK1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9296697-B2 Hetaryl-substituted guanidine compounds and use thereof as binding partners for 5-HT5-receptors ABBOTT LABORATORIES (US) 2016-03-29 US claimed