SCHEMBL176217

SCHEMBL176217

COC(=O)[C@H]1CC[C@H](c2nc(-c3ccc(Nc4ccc(OC(F)(F)F)cc4)cc3)no2)CC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN10A Q9Y5Y9 1/20 0.51
ALDH1A1 P00352 3/20 0.47
MAPT P10636 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
POLB P06746 1/20 0.46
MAPK1 P28482 1/20 0.46
CHRNA7 P36544 6/20 0.44
PKM P14618 1/20 0.44
XBP1 P17861 1/20 0.44
GAA P10253 2/20 0.43
KDM4E B2RXH2 1/20 0.43
LMNA P02545 1/20 0.43
HTT P42858 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
AOC3 Q16853 2/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
TUBB4A P04350 1/20 0.42
TUBB P07437 1/20 0.42
TUBA3C P0DPH7 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30584896 0.83 ALDH1A1 (0.58) ALDH1A1MAPTSMN1; SMN2POLBMAPK1
SCHEMBL176218 0.83 SCN10A (0.45) SCN10AALDH1A1MAPTSMN1; SMN2POLB
SCHEMBL162574 0.81 SCN10A (0.49) SCN10AALDH1A1MAPTSMN1; SMN2POLB
SCHEMBL162488 0.81 SCN10A (0.49) SCN10AALDH1A1MAPTSMN1; SMN2POLB
SCHEMBL4529235 0.78 CYP1A2 (0.60) ALDH1A1MAPTSMN1; SMN2POLBGAA
SCHEMBL4529230 0.78 CYP1A2 (0.60) ALDH1A1MAPTSMN1; SMN2POLBGAA
SCHEMBL174317 0.75 S1PR4 (0.49) ALDH1A1MAPTSMN1; SMN2POLBGAA
SCHEMBL174328 0.75 S1PR4 (0.49) ALDH1A1MAPTSMN1; SMN2POLBGAA
SCHEMBL24844551 0.74 NR1H4 (0.60) SMN1; SMN2GAALMNAHTTAOC3
SCHEMBL30584793 0.74 ALDH1A1 (0.56) ALDH1A1MAPTSMN1; SMN2POLBMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2611783-A2 HETEROCYCLIC COMPOUNDS AS DGAT1 INHIBITORS Piramal Enterprises Limited (IN) 2013-07-10 EP disclosed
WO-2012029032-A2 HETEROCYCLIC COMPOUNDS AS DGAT1 INHIBITORS PIRAMAL LIFE SCIENCES LIMITED (IN) 2012-03-08 WO disclosed