SCHEMBL17623239

SCHEMBL17623239

C/C=C\c1ncnc(OC)c1C

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 1/20 0.34
EGFR P00533 1/20 0.32
CYP3A4 P08684 2/20 0.31
LMNA P02545 1/20 0.31
TP53 P04637 1/20 0.31
TSHR P16473 1/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HSD17B10 Q99714 1/20 0.31
HMGCR P04035 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24344447 0.80 PDPK1 (0.36) PDPK1ALDH1A1HSD17B10
SCHEMBL19724521 0.79 APLNR (0.30)
SCHEMBL6796490 0.76 PDPK1 (0.45) PDPK1LMNATSHRALDH1A1HSD17B10
SCHEMBL16091312 0.72 LIMK1 (0.36) EGFR
SCHEMBL17623236 0.72 CNR2 (0.31) KDM4EALDH1A1
SCHEMBL12051534 0.70 PDPK1 (0.41) PDPK1LMNATSHRALDH1A1HSD17B10
SCHEMBL19215165 0.70
SCHEMBL179602 0.67 LIMK1 (0.38) PDPK1LMNATP53ALDH1A1HSD17B10
SCHEMBL179607 0.67 PDPK1 (0.38) PDPK1TSHRALDH1A1HSD17B10
SCHEMBL23717803 0.67 PDPK1 (0.38) PDPK1CYP3A4TSHRALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016044641-A2 CARM1 INHIBITORS AND USES THEREOF Epizyme, Inc. (US) 2016-03-24 WO disclosed