SCHEMBL17640586

SCHEMBL17640586

COC(=O)[C@H](CP)NC(=O)[C@H](CC(C)C)NC(=O)OC(C)(C)C

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CTSL P07711 2/20 0.56
CTSB P07858 1/20 0.56
CTSS P25774 1/20 0.56
CTSK P43235 1/20 0.56
CAPN1 P07384 1/20 0.50
REN P00797 2/20 0.46
GAA P10253 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
AAK1 Q2M2I8 1/20 0.46
BIRC2 Q13490 1/20 0.44
PSEN1 P49768 3/20 0.43
PSEN2 P49810 3/20 0.43
APH1B Q8WW43 3/20 0.43
NCSTN Q92542 3/20 0.43
APH1A Q96BI3 3/20 0.43
PSENEN Q9NZ42 3/20 0.43
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA7 P43166 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17640589 0.94 CTSK (0.51) CTSLCTSBCTSSCTSKCAPN1
SCHEMBL1176795 0.92 CTSL (0.62) CTSLCTSBCTSSCTSKCAPN1
SCHEMBL1026994 0.92 CTSL (0.62) CTSLCTSBCTSSCTSKCAPN1
SCHEMBL1026997 0.92 CTSL (0.62) CTSLCTSBCTSSCTSKCAPN1
SCHEMBL4576576 0.89 CTSL (0.56) CTSLCTSBCTSSCTSKCAPN1
SCHEMBL2632711 0.88 CTSL (0.58) CTSLCTSBCTSSCTSKCAPN1
SCHEMBL24130602 0.86 CTSL (0.60) CTSLCTSBCTSSCTSKCAPN1
SCHEMBL18762521 0.86 CTSL (0.53) CTSLCTSBCTSSCTSKCAPN1
SCHEMBL28948914 0.86 CTSL (0.56) CTSLCTSBCTSSCTSKCAPN1
SCHEMBL26818450 0.86 CTSL (0.56) CTSLCTSBCTSSCTSKCAPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016046843-A1 PROCESS FOR THE PREPARATION OF (S)-4-METHYL-N-((S)-1-(((S)-4-METHYL-1-((R)-2-METHYLOXIRAN-2-YL)-1-OXO PENTAN-2-YL) AMINO)-1-OXO-3-PHENYLPROPAN-2-YL)-2-((S)-2-(2-MORPHOLINOACETAMIDO)-4-PHENYLBUTANAMIDO) PENTANAMIDE BIOPHORE INDIA PHARMACEUTICALS PVT. LTD. (IN) 2016-03-31 WO disclosed