SCHEMBL1764208

SCHEMBL1764208

CC(NC(=O)OCc1ccccc1)P(=O)(O)CC(Cc1ccc(-c2ccccc2)cc1)C(=O)O

nearest known ligand 0.70

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ACE2 Q9BYF1 1/20 0.69
ECE1 P42892 12/20 0.61
MME P08473 11/20 0.61
MMP2 P08253 1/20 0.57
MMP9 P14780 1/20 0.57
MMP8 P22894 1/20 0.57
MMP14 P50281 1/20 0.57
MMP1 P03956 1/20 0.56
MMP3 P08254 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7613489 1.00 ACE2 (0.69) ACE2ECE1MMEMMP2MMP9
SCHEMBL24991304 1.00 ACE2 (0.69) ACE2ECE1MMEMMP2MMP9
SCHEMBL7613146 1.00 ACE2 (0.69) ACE2ECE1MMEMMP2MMP9
SCHEMBL6923615 0.92 ACE2 (0.58) ACE2ECE1MMEMMP2MMP9
SCHEMBL7619363 0.91 ACE2 (0.68) ACE2ECE1MMEMMP2MMP9
SCHEMBL7619360 0.91 ACE2 (0.68) ACE2ECE1MMEMMP2MMP9
SCHEMBL7620840 0.91 ACE2 (0.68) ACE2ECE1MMEMMP2MMP9
SCHEMBL7615297 0.88 ECE1 (0.76) ACE2ECE1MME
SCHEMBL6928872 0.88 ACE2 (0.66) ACE2ECE1MMEMMP2MMP9
SCHEMBL7611003 0.85 ANPEP (0.54) ACE2MME

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10131681-B2 Aminophosphinic derivatives that can be used in the treatment of pain PHARMALEADS (FR) 2018-11-20 US disclosed
US-20140161839-A1 AMINOPHOSPHINIC DERIVATIVES THAT CAN BE USED IN THE TREATMENT OF PAIN PHARMALEADS (FR) 2014-06-12 US disclosed
US-8703747-B2 Aminophosphinic derivatives that can be used in the treatment of pain PHARMALEADS (FR) 2014-04-22 US disclosed
US-20110124601-A1 AMINOPHOSPHINIC DERIVATIVES THAT CAN BE USED IN THE TREATMENT OF PAIN PHARMALEADS 2011-05-26 US disclosed
EP-1073664-B1 (ALPHA-AMINOPHOSPHINO) PEPTIDESDERIVATIVE AND COMPOSITIONS CONTAINING SAME INST NAT SANTE RECH MED (FR) 2002-10-23 EP disclosed
EP-1009750-B1 NOVEL (ALPHA-AMINOPHOSPHINO) PEPTIDE DERIVATIVES, METHOD FOR MAKING SAME AND THERAPEUTIC APPLICATIONS THEREOF INST NAT SANTE RECH MED (FR) 2002-07-31 EP disclosed
US-6391866-B1 ANALGESICS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2002-05-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110124601-A1 AMINOPHOSPHINIC DERIVATIVES THAT CAN BE USED IN THE TREATMENT OF PAIN OPRM1, HRH3, HRH4 ACE2 3562/4885ECE1 4157/4885MME 3670/4885
US-10131681-B2 Aminophosphinic derivatives that can be used in the treatment of pain OPRM1, HRH3, HRH4 ACE2 3454/4885ECE1 4097/4885MME 3490/4885
US-20140161839-A1 AMINOPHOSPHINIC DERIVATIVES THAT CAN BE USED IN THE TREATMENT OF PAIN OPRM1, HRH3, HRH4 ACE2 3454/4885ECE1 4097/4885MME 3490/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.