SCHEMBL17643170

SCHEMBL17643170

O=c1[nH]c2c(ccc3ncccc32)c(=O)o1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NCOA1 Q15788 2/20 0.49
MAPT P10636 2/20 0.46
KDM4E B2RXH2 1/20 0.46
F2 P00734 1/20 0.45
CFD P00746 1/20 0.45
CYP1A2 P05177 2/20 0.44
CYP1B1 Q16678 2/20 0.44
CYP1A1 P04798 1/20 0.42
CYP3A4 P08684 1/20 0.39
NCOA3 Q9Y6Q9 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
CYP19A1 P11511 3/20 0.38
LMNA P02545 2/20 0.38
MEN1 O00255 1/20 0.38
HSP90AA1 P07900 1/20 0.38
HSP90AB1 P08238 1/20 0.38
HTT P42858 1/20 0.38
BLM P54132 1/20 0.38
KMT2A Q03164 1/20 0.38
HIF1A Q16665 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17643178 0.77 MAPT (0.54) MAPTKDM4EF2CFDCYP1A2
SCHEMBL1522777 0.75 PARP1 (0.53) F2CFDHTTAURKAPARP1
SCHEMBL2098564 0.73 MCL1 (0.67) MAPTKDM4EF2CFDSMN1; SMN2
SCHEMBL21658311 0.71 F2 (0.55) MAPTF2CFDCYP1A2SMN1; SMN2
SCHEMBL29832015 0.70 KIF11 (0.55) MAPTKDM4ECYP1A2CYP3A4SMN1; SMN2
SCHEMBL458963 0.70 KIF11 (0.55) MAPTKDM4ECYP1A2CYP3A4SMN1; SMN2
SCHEMBL22650664 0.70 MAPT (0.47) NCOA1MAPTKDM4ECYP1A2CYP1B1
SCHEMBL1416592 0.69 MAPT (0.50) NCOA1MAPTKDM4ECYP1A2CYP1B1
SCHEMBL660137 0.69 MAPT (0.50) NCOA1MAPTKDM4ECYP1A2CYP1B1
SCHEMBL26675637 0.69 PARP1 (0.51) MAPTKDM4ECYP3A4SMN1; SMN2CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3197982-B1 MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2020-05-06 EP disclosed
US-10544360-B2 Materials for organic electroluminescent devices MERCK PATENT GMBH (DE) 2020-01-28 US disclosed
WO-2016045765-A1 MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2016-03-31 WO disclosed