SCHEMBL17644608

SCHEMBL17644608

BrC1(c2ccccc2)C#C1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 3/20 0.39
OPRK1 P41145 2/20 0.39
OPRL1 P41146 2/20 0.39
LMNA P02545 1/20 0.33
TSHR P16473 1/20 0.33
ALOX12 P18054 1/20 0.33
ACHE P22303 1/20 0.33
ALDH1A1 P00352 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
MAOB P27338 5/20 0.32
MAOA P21397 4/20 0.32
PNMT P11086 1/20 0.32
TAAR1 Q96RJ0 1/20 0.32
MEN1 O00255 1/20 0.31
CYP2C9 P11712 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16266151 0.69 OPRM1 (0.36) OPRM1OPRK1OPRL1ALDH1A1MAOB
SCHEMBL2969527 0.65 OPRM1 (0.44) OPRM1OPRK1OPRL1MAOBMAOA
SCHEMBL11453348 0.65 ALDH1A1 (0.40) OPRM1OPRK1OPRL1LMNATSHR
SCHEMBL15327787 0.65 MEN1 (0.35) OPRM1OPRK1OPRL1TSHRMAOB
SCHEMBL10876622 0.63 OPRM1 (0.41) OPRM1OPRK1OPRL1LMNAALDH1A1
SCHEMBL5480380 0.63 OPRM1 (0.41) OPRM1OPRK1OPRL1ALDH1A1MAOB
SCHEMBL5076533 0.63 MEN1 (0.39) OPRM1OPRK1OPRL1MAOBMAOA
SCHEMBL968174 0.61 HDAC4 (0.42) OPRM1OPRK1OPRL1MAOBMAOA
SCHEMBL15954140 0.61 DPP4 (0.41) OPRM1OPRK1OPRL1MAOBMAOA
SCHEMBL5274478 0.61 ALDH1A1 (0.31) OPRM1OPRK1OPRL1LMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2782903-B1 NOVEL PYRROLIDINE DERIVATIVES AS INHIBITORS OF CATHEPSIN HOFFMANN LA ROCHE (CH) 2016-04-06 EP claimed