SCHEMBL17656261

SCHEMBL17656261

Brc1ccc(-c2cnc([C@H]3N[C@@H]4CC[C@H]3C4)[nH]2)cc1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAPK13 O15264 1/20 0.45
MAPK12 P53778 1/20 0.45
MAPK11 Q15759 1/20 0.45
MAPK14 Q16539 1/20 0.45
TRPV1 Q8NER1 1/20 0.37
SSTR3 P32745 14/20 0.36
KCNH2 Q12809 13/20 0.36
CACNA1F O60840 2/20 0.36
CACNA1D Q01668 2/20 0.36
CACNA1S Q13698 2/20 0.36
CACNA1C Q13936 2/20 0.36
PTGES O14684 1/20 0.35
HPGDS O60760 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17656297 0.88 MAPK13 (0.36) MAPK13MAPK12MAPK11MAPK14SSTR3
SCHEMBL12437629 0.83 SSTR3 (0.36) SSTR3KCNH2CACNA1FCACNA1DCACNA1S
SCHEMBL12436380 0.78 SSTR3 (0.33) MAPK13MAPK12MAPK11MAPK14SSTR3
SCHEMBL16891266 0.77 SSTR3 (0.34) SSTR3KCNH2CACNA1FCACNA1DCACNA1S
SCHEMBL10132664 0.76 MAPK13 (0.53) MAPK13MAPK12MAPK11MAPK14TRPV1
SCHEMBL825046 0.76 MAPK13 (0.53) MAPK13MAPK12MAPK11MAPK14TRPV1
SCHEMBL456621 0.75 MAPK13 (0.55) MAPK13MAPK12MAPK11MAPK14TRPV1
SCHEMBL9977194 0.75 MAPK13 (0.46) MAPK13MAPK12MAPK11MAPK14TRPV1
SCHEMBL16577375 0.75 MAPK13 (0.51) MAPK13MAPK12MAPK11MAPK14TRPV1
SCHEMBL17014411 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3002281-B1 ANTIVIRAL COMPOUNDS GILEAD PHARMASSET LLC (US) 2017-09-13 EP disclosed
EP-3002281-A1 ANTIVIRAL COMPOUNDS Gilead Pharmasset LLC (US) 2016-04-06 EP disclosed