SCHEMBL17656753

SCHEMBL17656753

O=C(O)c1ccc(CN2CCN(c3cccc(CO)c3)CC2)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 3/20 0.63
ITGA2B P08514 3/20 0.63
DRD2 P14416 2/20 0.58
DRD3 P35462 1/20 0.58
DRD4 P21917 1/20 0.54
HTR2A P28223 1/20 0.52
HTR2C P28335 1/20 0.52
HTR2B P41595 1/20 0.52
HTR7 P34969 2/20 0.52
HTR1A P08908 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.51
KDM4E B2RXH2 1/20 0.49
TP53 P04637 1/20 0.49
MAPT P10636 1/20 0.49
TSHR P16473 1/20 0.49
HSD17B10 Q99714 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
HIF1A Q16665 1/20 0.49
HDAC4 P56524 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12526363 0.85 DRD2 (0.56) ITGB3ITGA2BDRD2DRD3DRD4
SCHEMBL4021071 0.84 DRD2 (0.68) ITGB3ITGA2BDRD2DRD3DRD4
Hydrochloric Acid SCHEMBL10713081 0.84 DRD4 (0.68) ITGB3ITGA2BDRD2DRD3DRD4
SCHEMBL1066467 0.82 HTR2A (0.72) ITGB3ITGA2BDRD4HTR2AHTR2C
Hydrochloric Acid SCHEMBL4653252 0.81 HTR2A (0.71) ITGB3ITGA2BDRD4HTR2AHTR2C
SCHEMBL27519383 0.80 HDAC4 (0.71) SMN1; SMN2KDM4EMAPTTSHRCYP2D6
SCHEMBL17656756 0.79 AOC3 (0.55) DRD2DRD3DRD4TSHRHSD17B10
SCHEMBL31593043 0.79 CYP2D6 (0.69) ITGB3ITGA2BDRD2DRD3DRD4
SCHEMBL27040086 0.79 CYP2D6 (0.69) ITGB3ITGA2BDRD2DRD3DRD4
SCHEMBL10074441 0.78 HDAC1 (0.62) SMN1; SMN2KDM4EMAPTCYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2695881-B1 GUANIDINE COMPOUND ASTELLAS PHARMA INC (JP) 2016-04-27 EP disclosed
EP-3002278-A1 GUANIDINE COMPOUND Astellas Pharma Inc. (JP) 2016-04-06 EP disclosed