SCHEMBL17667274

SCHEMBL17667274

CN(C(=O)OC(C)(C)C)[C@@H]1CCCN(c2nc(Cl)nc3c2CCCC3)C1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SPR P35270 1/20 0.43
PDE10A Q9Y233 1/20 0.41
RET P07949 1/20 0.39
KIF18A Q8NI77 1/20 0.39
HSD11B1 P28845 1/20 0.36
AAK1 Q2M2I8 1/20 0.36
PRKDC P78527 2/20 0.36
HRH4 Q9H3N8 3/20 0.35
GBA1 P04062 2/20 0.34
JAK3 P52333 3/20 0.33
BTK Q06187 2/20 0.33
KDM4D Q6B0I6 1/20 0.33
TP53 P04637 1/20 0.33
GLA P06280 1/20 0.33
JAK2 O60674 1/20 0.33
LCK P06239 1/20 0.33
TRPV1 Q8NER1 1/20 0.32
PIK3CD O00329 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17667288 0.98 SPR (0.45) SPRPDE10ARETKIF18AHSD11B1
SCHEMBL17628270 0.95 SPR (0.46) SPRPDE10ARETKIF18AHSD11B1
SCHEMBL17628272 0.95 SPR (0.46) SPRPDE10ARETKIF18AHSD11B1
SCHEMBL17627935 0.86 PRKDC (0.39) PRKDCHRH4GBA1JAK3BTK
SCHEMBL17628075 0.83 PRKDC (0.39) SPRPRKDCHRH4GBA1JAK3
SCHEMBL17628208 0.83 CFTR (0.42) SPRPDE10AHSD11B1AAK1HRH4
SCHEMBL17628211 0.83 CFTR (0.42) SPRPDE10AHSD11B1AAK1HRH4
SCHEMBL17667302 0.81 HRH4 (0.36) PRKDCHRH4GBA1TP53GLA
SCHEMBL17667301 0.81 HRH4 (0.36) PRKDCHRH4GBA1TP53GLA
SCHEMBL17667275 0.79 HRH4 (0.35) PRKDCHRH4GBA1JAK3TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3006439-A1 BICYCLIC DERIVATIVE CONTAINING PYRIMIDINE RING, AND PREPARATION METHOD THEREFOR Yuhan Corporation (KR) 2016-04-13 EP disclosed