SCHEMBL17672811

SCHEMBL17672811

N#Cc1ccc(C#Cc2ccc(O)cc2F)c(F)c1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.47
CA2 P00918 1/20 0.47
CA3 P07451 1/20 0.47
CA6 P23280 1/20 0.47
CA9 Q16790 1/20 0.47
CA14 Q9ULX7 1/20 0.47
CYP19A1 P11511 3/20 0.43
MMP3 P08254 1/20 0.42
AR P10275 4/20 0.41
ESR1 P03372 5/20 0.41
ESR2 Q92731 5/20 0.41
FFAR1 O14842 1/20 0.39
FFAR4 Q5NUL3 1/20 0.39
TRPV4 Q9HBA0 1/20 0.39
HAO1 Q9UJM8 2/20 0.38
CYP11B1 P15538 1/20 0.37
CYP11B2 P19099 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17672698 0.91 CA12 (0.50) CA12CA2CA3CA6CA9
SCHEMBL17672970 0.91 CA12 (0.50) CA12CA2CA3CA6CA9
SCHEMBL17672587 0.89 MRGPRX4 (0.42) CA12CA2CA3CA6CA9
SCHEMBL17672545 0.89 MRGPRX4 (0.42) CA12CA2CA3CA6CA9
SCHEMBL17672810 0.86 AR (0.49) CA12CA2CA3CA6CA9
SCHEMBL17672734 0.85 MAOB (0.40) CA12CA2CA3CA6CA9
4-Cyanophenol SCHEMBL6894396 0.84 CA9 (0.59) CA12CA2CA3CA6CA9
SCHEMBL176946 0.81 TRPV4 (0.57) ARESR1ESR2TRPV4CYP11B1
SCHEMBL16182684 0.79 APP (0.47) CA12CA2CA3CA6CA9
SCHEMBL31122790 0.79 TRPV4 (0.55) ARESR1ESR2TRPV4CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016055947-A1 ALKYNE COMPOUNDS AS S-NITROSOGLUTATHIONE REDUCTASE INHIBITORS GLENMARK PHARMACEUTICALS S.A. (CH) 2016-04-14 WO disclosed
WO-2016055947-A1 ALKYNE COMPOUNDS AS S-NITROSOGLUTATHIONE REDUCTASE INHIBITORS GLENMARK PHARMACEUTICALS S.A. (CH) 2016-04-14 WO disclosed