SCHEMBL17673155

SCHEMBL17673155

O=[N+]([O-])c1ccn[c]c1F

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 4/20 0.38
ATM Q13315 1/20 0.38
ALDH1A1 P00352 3/20 0.37
HIF1A Q16665 2/20 0.37
VCAM1 P19320 1/20 0.35
HTT P42858 1/20 0.35
RAB9A P51151 1/20 0.35
PDE10A Q9Y233 1/20 0.34
POLB P06746 2/20 0.34
MAPT P10636 2/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
CASP6 P55212 2/20 0.34
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
THRB P10828 1/20 0.34
PKM P14618 1/20 0.34
IDO1 P14902 1/20 0.34
RECQL P46063 1/20 0.34
TDO2 P48775 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10767704 0.80 TDP1 (0.39) TDP1ALDH1A1VCAM1HTTPDE10A
SCHEMBL3200434 0.76 TDP1 (0.38) TDP1ALDH1A1PDE10APOLBMAPT
SCHEMBL12274556 0.72 CASP6 (0.41) TDP1ALDH1A1CASP6KDM4ELMNA
SCHEMBL2067226 0.72 ALDH1A1 (0.42) TDP1ALDH1A1HTTMAPTMEN1
SCHEMBL29241423 0.67 TDP1 (0.45) TDP1ATMALDH1A1HIF1AVCAM1
SCHEMBL6401677 0.66
SCHEMBL407098 0.66
SCHEMBL2602388 0.65 ALDH1A1 (0.50) TDP1ATMALDH1A1HIF1AVCAM1
SCHEMBL2075134 0.65 TDP1 (0.45) TDP1ATMALDH1A1HIF1AVCAM1
SCHEMBL3200439 0.64 ALDH1A1 (0.34) TDP1ALDH1A1HTTPOLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3204360-A1 THERAPEUTIC COMPOUNDS AND USES THEREOF Genentech, Inc. (US) 2017-08-16 EP disclosed
WO-2016055028-A1 THERAPEUTIC COMPOUNDS AND USES THEREOF GENENTECH, INC. (US) 2016-04-14 WO disclosed