SCHEMBL17675170

SCHEMBL17675170

CCc1ccnc(NC(=O)c2ccc(Oc3ncnc4ccc([N+](=O)[O-])cc34)cc2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.53
BTK Q06187 2/20 0.53
ERBB2 P04626 1/20 0.53
TEC P42680 1/20 0.53
TXK P42681 1/20 0.53
BLK P51451 1/20 0.53
BMX P51813 1/20 0.53
JAK3 P52333 1/20 0.53
ERBB4 Q15303 1/20 0.53
KDR P35968 1/20 0.46
MAPT P10636 6/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
ALDH1A1 P00352 2/20 0.44
HTT P42858 1/20 0.44
KMT2A Q03164 3/20 0.43
USP2 O75604 1/20 0.43
MEN1 O00255 1/20 0.42
MMP13 P45452 1/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17675493 0.88 BTK (0.68) EGFRBTKERBB2TECTXK
SCHEMBL17675208 0.86 BTK (0.56) EGFRBTKERBB2TECTXK
SCHEMBL17675311 0.85 BTK (0.66) EGFRBTKKDRMAPTALDH1A1
SCHEMBL17675293 0.84 EGFR (0.49) EGFRBTKKDRMAPTKMT2A
SCHEMBL17675440 0.83 BTK (0.55) EGFRBTKERBB2TECTXK
SCHEMBL17675213 0.81 EGFR (0.79) EGFRBTKERBB2TECTXK
SCHEMBL17675511 0.76 KMT2A (0.55) EGFRBTKERBB2TECTXK
SCHEMBL17675289 0.73 BTK (0.72) EGFRBTKERBB2TECTXK
SCHEMBL17675318 0.73 BTK (0.66) EGFRBTKERBB2TECTXK
SCHEMBL17675515 0.72 BTK (0.49) EGFRBTKERBB2TECTXK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016055982-A1 QUINOLINE AND QUINAZOLINE COMPOUNDS ACERTA PHARMA B.V. (NL) 2016-04-14 WO disclosed