SCHEMBL17675440

SCHEMBL17675440

CCc1ccnc(NC(=O)c2ccc(Oc3cnnc4ccc([N+](=O)[O-])cc34)cc2)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BTK Q06187 7/20 0.55
EGFR P00533 6/20 0.55
ERBB2 P04626 1/20 0.55
TEC P42680 1/20 0.55
TXK P42681 1/20 0.55
BLK P51451 1/20 0.55
BMX P51813 1/20 0.55
JAK3 P52333 1/20 0.55
ERBB4 Q15303 1/20 0.55
PDGFRA P16234 2/20 0.42
KDR P35968 2/20 0.42
MAPT P10636 3/20 0.41
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
MMP13 P45452 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
NPC1 O15118 1/20 0.41
PKM P14618 1/20 0.41
RAB9A P51151 1/20 0.41
USP2 O75604 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17675493 0.90 BTK (0.68) BTKEGFRERBB2TECTXK
SCHEMBL17675205 0.86 BTK (0.58) BTKEGFRERBB2TECTXK
SCHEMBL17675170 0.83 EGFR (0.53) BTKEGFRERBB2TECTXK
SCHEMBL17675197 0.82 EGFR (0.82) BTKEGFRERBB2TECTXK
SCHEMBL17683792 0.80 EGFR (0.66) BTKEGFRERBB2TECTXK
SCHEMBL17675511 0.78 KMT2A (0.55) BTKEGFRERBB2TECTXK
SCHEMBL17675318 0.75 BTK (0.66) BTKEGFRERBB2TECTXK
SCHEMBL17675289 0.75 BTK (0.72) BTKEGFRERBB2TECTXK
SCHEMBL17675515 0.74 BTK (0.49) BTKEGFRERBB2TECTXK
SCHEMBL17675288 0.72 MAPT (0.48) BTKEGFRERBB2TECTXK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016055982-A1 QUINOLINE AND QUINAZOLINE COMPOUNDS ACERTA PHARMA B.V. (NL) 2016-04-14 WO disclosed