SCHEMBL17675301

SCHEMBL17675301

Nc1ccc2nccc(Oc3ccc(C(=O)Nc4ccccn4)nc3)c2c1

nearest known ligand 0.58

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BTK Q06187 10/20 0.58
EGFR P00533 7/20 0.55
CYP3A4 P08684 1/20 0.50
KDR P35968 1/20 0.50
AXL P30530 1/20 0.49
MET P08581 6/20 0.49
GRM5 P41594 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17675235 0.88 BTK (0.73) BTKEGFRCYP3A4KDR
SCHEMBL17675399 0.85 BTK (0.81) BTKEGFRCYP3A4KDRAXL
SCHEMBL17675471 0.85 BTK (0.52) BTKEGFRCYP3A4KDRAXL
SCHEMBL17675237 0.83 EGFR (0.80) BTKEGFRCYP3A4KDRAXL
SCHEMBL17675239 0.78 BTK (0.82) BTKEGFRCYP3A4KDRAXL
SCHEMBL17675303 0.76 BTK (0.70) BTKEGFRCYP3A4KDR
SCHEMBL17675438 0.75 BTK (0.59) BTKEGFR
SCHEMBL17675336 0.74 BTK (0.63) BTKEGFRCYP3A4KDRAXL
SCHEMBL17683824 0.74 BTK (1.00) BTKEGFRCYP3A4KDRAXL
SCHEMBL17675332 0.73 BTK (0.70) BTKEGFRKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016055982-A1 QUINOLINE AND QUINAZOLINE COMPOUNDS ACERTA PHARMA B.V. (NL) 2016-04-14 WO disclosed
WO-2016055982-A1 QUINOLINE AND QUINAZOLINE COMPOUNDS ACERTA PHARMA B.V. (NL) 2016-04-14 WO disclosed