SCHEMBL17675433

SCHEMBL17675433

COc1cc2ncnc(Oc3ccc(C(=O)Nc4cc(C(F)(F)F)ccn4)cc3)c2cc1N

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 11/20 0.59
BRAF P15056 8/20 0.55
MAPK14 Q16539 2/20 0.55
TNNI3K Q59H18 2/20 0.55
RAF1 P04049 4/20 0.48
PDGFRA P16234 1/20 0.48
PDGFRB P09619 1/20 0.47
FLT4 P35916 1/20 0.47
CLK2 P49760 1/20 0.47
IRAK1 P51617 1/20 0.47
NEK4 P51957 1/20 0.47
MAP4K2 Q12851 1/20 0.47
HIPK4 Q8NE63 1/20 0.47
SRPK1 Q96SB4 1/20 0.47
CLK4 Q9HAZ1 1/20 0.47
MKNK2 Q9HBH9 1/20 0.47
MAP3K20 Q9NYL2 1/20 0.47
STK17A Q9UEE5 1/20 0.47
MAP4K5 Q9Y4K4 1/20 0.47
GRM5 P41594 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17683793 0.94 KDR (0.54) KDRBRAFMAPK14TNNI3KRAF1
SCHEMBL17683762 0.86 BTK (0.62) KDRBRAFMAPK14TNNI3KRAF1
SCHEMBL17675462 0.85 BTK (0.51) KDRBRAFMAPK14TNNI3KCLK2
SCHEMBL17675474 0.85 BTK (0.60) KDRBRAFPDGFRAPDGFRBFLT4
SCHEMBL17675293 0.79 EGFR (0.49) KDRBRAFMAPK14TNNI3KPDGFRB
SCHEMBL17675352 0.77 EGFR (0.74) KDRBRAFMAPK14TNNI3KGRM5
SCHEMBL17675531 0.77 BTK (0.59) KDRPDGFRAMET
SCHEMBL1781683 0.76 BRAF (0.84) KDRBRAFMAPK14TNNI3KRAF1
SCHEMBL17675216 0.74 BTK (0.54) KDRBRAFMAPK14TNNI3KCLK2
SCHEMBL17675203 0.74 BTK (0.73) KDRPDGFRAMET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016055982-A1 QUINOLINE AND QUINAZOLINE COMPOUNDS ACERTA PHARMA B.V. (NL) 2016-04-14 WO disclosed