SCHEMBL1767591

SCHEMBL1767591

Cn1cc(C(=O)Nc2ccc(F)cc2-c2ccc(Cl)cc2)c(C(F)F)n1.Cn1cc(C(=O)Nc2ccc(F)cc2-c2cccc(Cl)c2)c(C(F)F)n1.Cn1cc(C(=O)Nc2ccccc2-c2ccc(Cl)cc2)c(C(F)F)n1

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 10/20 0.46
SUCNR1 Q9BXA5 2/20 0.43
TDP1 Q9NUW8 1/20 0.43
CHRM2 P08172 2/20 0.42
CHRM1 P11229 2/20 0.42
JAK2 O60674 3/20 0.42
JAK1 P23458 1/20 0.42
F10 P00742 1/20 0.42
NTRK1 P04629 1/20 0.41
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1134824 0.93 CHRM3 (0.51) CHRM3CHRM2CHRM1JAK2JAK1
SCHEMBL302468 0.91 JAK2 (0.48) CHRM3TDP1CHRM1JAK2JAK1
SCHEMBL1134849 0.90 CHRM3 (0.49) CHRM3CHRM2CHRM1
SCHEMBL121957 0.88 TDP1 (0.53) CHRM3SUCNR1TDP1F10NTRK1
SCHEMBL29419144 0.88 TDP1 (0.53) CHRM3SUCNR1TDP1F10NTRK1
SCHEMBL13491718 0.86 CHRM3 (0.50) CHRM3CHRM2CHRM1NTRK1MAPT
SCHEMBL303819 0.85 CHRM3 (0.48) CHRM3JAK2JAK1NTRK1MAPT
SCHEMBL20875262 0.84 NTRK1 (0.52) CHRM3TDP1NTRK1MAPT
SCHEMBL1136276 0.84 CHRM3 (0.51) CHRM3CHRM2CHRM1
SCHEMBL304216 0.84 SSTR2 (0.45) CHRM3SUCNR1TDP1JAK2JAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2496560-A1 PROCESS FOR PREPARING 1,3-DISUBSTITUTED PYRAZOLE COMPOUNDS BASF SE (DE) 2012-09-12 EP disclosed
EP-2496561-A1 PROCESS FOR PREPARING AMINALE AND THEIR USE FOR PREPARING 1,3-DISUBSTITUTED PYRAZOLE COMPOUNDS BASF SE (DE) 2012-09-12 EP disclosed
WO-2011054732-A1 PROCESS FOR PREPARING 1,3-DISUBSTITUTED PYRAZOLE COMPOUNDS BASF SE (DE) 2011-05-12 WO disclosed
WO-2011054733-A1 PROCESS FOR PREPARING AMINALE AND THEIR USE FOR PREPARING 1,3-DISUBSTITUTED PYRAZOLE COMPOUNDS BASF SE (DE) 2011-05-12 WO disclosed