SCHEMBL1767993

SCHEMBL1767993

CN(C)C(=O)c1nc(N)nc2ccc(C3(C)CCC3)cc12

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 9/20 0.44
AKT1 P31749 3/20 0.37
HSP90AB1 P08238 2/20 0.37
SCN10A Q9Y5Y9 1/20 0.33
AKT2 P31751 2/20 0.32
NUDT1 P36639 1/20 0.32
ALDH1A1 P00352 1/20 0.32
ADORA3 P0DMS8 2/20 0.32
MAP4K1 Q92918 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1767995 0.87 HSP90AA1 (0.46) HSP90AA1HSP90AB1SCN10AALDH1A1
SCHEMBL12273557 0.87 HSP90AA1 (0.50) HSP90AA1AKT1HSP90AB1AKT2
SCHEMBL1767930 0.87 HSP90AA1 (0.44) HSP90AA1HSP90AB1SCN10A
SCHEMBL1768050 0.85 HSP90AA1 (0.45) HSP90AA1ALDH1A1
SCHEMBL12273696 0.81 HSP90AA1 (0.68) HSP90AA1AKT1HSP90AB1NUDT1ALDH1A1
SCHEMBL12273083 0.81 HSP90AA1 (0.49) HSP90AA1
SCHEMBL12273050 0.75 HSP90AA1 (0.52) HSP90AA1HSP90AB1ALDH1A1
SCHEMBL12273344 0.75 HSP90AA1 (0.50) HSP90AA1HSP90AB1
Bicarbonate SCHEMBL1768007 0.74 EGLN1 (0.41) HSP90AA1HSP90AB1NUDT1ALDH1A1
SCHEMBL16271130 0.74 HSP90AA1 (0.39) HSP90AA1HSP90AB1NUDT1ADORA3MAP4K1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2504314-A1 QUINAZOLINE DERIVATIVES Merck Patent GmbH (DE) 2012-10-03 EP disclosed
WO-2011060873-A1 QUINAZOLINE DERIVATIVES MERCK PATENT GMBH (DE) 2011-05-26 WO disclosed