SCHEMBL1767995

SCHEMBL1767995

CCN(CC)C(=O)c1nc(N)nc2ccc(C3(C)CCC3)cc12

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 8/20 0.46
ALDH1A1 P00352 2/20 0.36
HPGD P15428 2/20 0.36
LMNA P02545 1/20 0.36
DHFR P00374 1/20 0.35
HSP90AB1 P08238 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
SCN10A Q9Y5Y9 1/20 0.33
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12273050 0.88 HSP90AA1 (0.52) HSP90AA1ALDH1A1HPGDLMNADHFR
SCHEMBL1767993 0.87 HSP90AA1 (0.44) HSP90AA1ALDH1A1HSP90AB1SCN10A
SCHEMBL1767930 0.86 HSP90AA1 (0.44) HSP90AA1DHFRHSP90AB1SCN10A
SCHEMBL12273754 0.83 HSP90AA1 (0.49) HSP90AA1ALDH1A1DHFRSLC6A4
SCHEMBL12273492 0.83 HSP90AA1 (0.67) HSP90AA1ALDH1A1HPGDLMNADHFR
SCHEMBL1768050 0.82 HSP90AA1 (0.45) HSP90AA1ALDH1A1HPGDMEN1KMT2A
SCHEMBL3088463 0.78 HSP90AA1 (0.53) HSP90AA1ALDH1A1HPGDLMNADHFR
SCHEMBL3087968 0.77 HSP90AA1 (0.47) HSP90AA1ALDH1A1HPGDLMNADHFR
SCHEMBL3088521 0.77 HSP90AB1 (0.45) ALDH1A1HPGDLMNAHSP90AB1SMN1; SMN2
SCHEMBL3092345 0.77 ALDH1A1 (0.41) ALDH1A1HPGDLMNADHFRMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2504314-A1 QUINAZOLINE DERIVATIVES Merck Patent GmbH (DE) 2012-10-03 EP disclosed
WO-2011060873-A1 QUINAZOLINE DERIVATIVES MERCK PATENT GMBH (DE) 2011-05-26 WO disclosed