SCHEMBL1768050

SCHEMBL1768050

CN(Cc1ccccc1)C(=O)c1nc(N)nc2ccc(C3(C)CCC3)cc12

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.45
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
PIN1 Q13526 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12273449 0.89 HSP90AA1 (0.51) HSP90AA1CYP3A4CYP2D6ALDH1A1HPGD
SCHEMBL1767930 0.86 HSP90AA1 (0.44) HSP90AA1CYP3A4CYP2D6
SCHEMBL1767993 0.85 HSP90AA1 (0.44) HSP90AA1ALDH1A1
SCHEMBL12273734 0.85 HSP90AA1 (0.49) HSP90AA1CYP3A4CYP2D6
SCHEMBL12448027 0.84 HSP90AA1 (0.66) HSP90AA1CYP3A4CYP2D6ALDH1A1HPGD
SCHEMBL1767995 0.82 HSP90AA1 (0.46) HSP90AA1ALDH1A1HPGDMEN1KMT2A
SCHEMBL13144830 0.80 CYP3A4 (0.48) CYP3A4CYP2D6ALDH1A1HPGDMEN1
SCHEMBL3099560 0.80 CYP3A4 (0.48) CYP3A4CYP2D6ALDH1A1HPGDMEN1
SCHEMBL3081057 0.79 CYP3A4 (0.53) CYP3A4CYP2D6MEN1KMT2A
Bicarbonate SCHEMBL16966267 0.78 CYP3A4 (0.43) CYP3A4CYP2D6ALDH1A1HPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2504314-A1 QUINAZOLINE DERIVATIVES Merck Patent GmbH (DE) 2012-10-03 EP disclosed
WO-2011060873-A1 QUINAZOLINE DERIVATIVES MERCK PATENT GMBH (DE) 2011-05-26 WO disclosed