SCHEMBL1768012

SCHEMBL1768012

CC(CCC(F)F)(CCC(F)F)c1ccc2c(c1)C(=O)C(=O)N2

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TGM2 P21980 5/20 0.44
CES1 P23141 4/20 0.43
ALDH1A1 P00352 1/20 0.42
MAOA P21397 8/20 0.40
MAOB P27338 8/20 0.40
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
CASP3 P42574 3/20 0.38
CAPN9 O14815 1/20 0.38
SLC6A11 P48066 1/20 0.38
PDE3B Q13370 1/20 0.38
PDE3A Q14432 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1767895 0.78 CES1 (0.38) TGM2CES1ALDH1A1MAOAMAOB
SCHEMBL30541907 0.76 TGM2 (0.55) TGM2CES1ALDH1A1MAOAMAOB
SCHEMBL1247409 0.76 TGM2 (0.55) TGM2CES1ALDH1A1MAOAMAOB
SCHEMBL2372316 0.73 CES1 (0.58) TGM2CES1ALDH1A1MAOAMAOB
SCHEMBL30120589 0.73 CES1 (0.58) TGM2CES1ALDH1A1MAOAMAOB
Hydrochloric Acid SCHEMBL11435666 0.71 CES1 (0.57) TGM2CES1ALDH1A1MAOAMAOB
SCHEMBL4202180 0.70 CES1 (0.56) TGM2CES1ALDH1A1MAOAMAOB
SCHEMBL13401353 0.70 TGM2 (0.55) TGM2CES1ALDH1A1MAOAMAOB
SCHEMBL9276654 0.68 TGM2 (0.42) TGM2CES1ALDH1A1MAOAMAOB
SCHEMBL2788213 0.68 MAOA (0.66) TGM2CES1ALDH1A1MAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2504314-A1 QUINAZOLINE DERIVATIVES Merck Patent GmbH (DE) 2012-10-03 EP disclosed
WO-2011060873-A1 QUINAZOLINE DERIVATIVES MERCK PATENT GMBH (DE) 2011-05-26 WO disclosed