SCHEMBL17680236

SCHEMBL17680236

CCc1cnc(N)c(OCC2CC2)c1

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 1/20 0.45
BRD4 O60885 1/20 0.41
CREBBP Q92793 1/20 0.41
CNR2 P34972 9/20 0.41
MAP4K3 Q8IVH8 2/20 0.40
DHFR P00374 1/20 0.39
CNR1 P21554 1/20 0.37
MAP3K12 Q12852 1/20 0.37
TRPC6 Q9Y210 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17681017 0.81 MAP4K4 (0.47) MAP4K4BRD4CREBBPCNR2MAP4K3
SCHEMBL19446090 0.80 CNR2 (0.40) CNR2CNR1TRPC6
SCHEMBL15880738 0.78 MAP4K4 (0.47) MAP4K4BRD4CREBBPCNR2MAP4K3
SCHEMBL19531672 0.77 DHFR (0.46) MAP4K4BRD4CREBBPCNR2MAP4K3
SCHEMBL91322 0.76 PTGS2 (0.48) DHFR
SCHEMBL15609364 0.74 MAP4K3 (0.50) MAP4K4MAP4K3
SCHEMBL19673294 0.73 BRD4 (0.39) BRD4CNR2
SCHEMBL18118645 0.73 EP300 (0.40) CNR2
SCHEMBL18400077 0.72 SCN9A (0.38) CNR2CNR1
SCHEMBL19446253 0.71 MAP3K12 (0.46) MAP3K12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016055028-A1 THERAPEUTIC COMPOUNDS AND USES THEREOF GENENTECH, INC. (US) 2016-04-14 WO disclosed