SCHEMBL1768416

SCHEMBL1768416

CC(C)(C)N(Cc1noc(-c2c3ccccc3nn2CCc2cccs2)n1)C(=O)O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.51
CYP2D6 P10635 2/20 0.51
SCN8A Q9UQD0 2/20 0.43
SCN1A P35498 1/20 0.37
SCN4A P35499 1/20 0.37
SCN5A Q14524 1/20 0.37
SCN9A Q15858 1/20 0.37
SCN2A Q99250 1/20 0.37
SCN3A Q9NY46 1/20 0.37
SCN10A Q9Y5Y9 1/20 0.37
HDAC3 O15379 1/20 0.36
HDAC4 P56524 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
ALDH1A1 P00352 4/20 0.34
MAPT P10636 4/20 0.34
LMNA P02545 2/20 0.34
KDM4E B2RXH2 1/20 0.34
GBA1 P04062 1/20 0.34
CRHBP P24387 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11896947 0.82 CYP1A2 (0.47) CYP1A2CYP2D6SCN8AALDH1A1MAPT
SCHEMBL11896946 0.82 CYP1A2 (0.54) CYP1A2CYP2D6SCN8ASCN1ASCN4A
SCHEMBL1768351 0.82 SCN8A (0.55) CYP1A2CYP2D6SCN8ASCN1ASCN4A
SCHEMBL1768182 0.81 CYP2D6 (0.72) CYP1A2CYP2D6SCN8ASCN1ASCN4A
SCHEMBL12649293 0.80 CYP1A2 (0.51) CYP1A2CYP2D6SCN8ASCN1ASCN4A
SCHEMBL1768208 0.80 SCN8A (0.52) CYP1A2CYP2D6SCN8ASCN1ASCN4A
SCHEMBL1768502 0.80 CYP1A2 (0.48) CYP1A2CYP2D6SCN8ASCN1ASCN4A
SCHEMBL1768415 0.78 CYP1A2 (0.43) CYP1A2CYP2D6SCN8ASCN1ASCN4A
SCHEMBL1768241 0.72 SCN8A (0.48) CYP1A2CYP2D6SCN8ASCN1ASCN4A
SCHEMBL1768484 0.68 CYP2D6 (0.47) CYP1A2CYP2D6SCN8ASCN1ASCN4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011061469-A1 INDAZOLE DERIVATIVES AND THEIR USE FOR BLOCKADING VOLTAGE DEPENDENT SODIUM CHANNELS UNIVERSITY COLLEGE LONDON (GB) 2011-05-26 WO disclosed