SCHEMBL17690495

SCHEMBL17690495

CC(C)(O)C#Cc1nc(Cl)n(Cc2ccc(C(F)(F)F)cc2)c1C(=O)NCc1ccc(-c2noc(=O)n2N)cc1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.37
PTGER4 P35408 5/20 0.36
PPARA Q07869 4/20 0.36
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36
CHRM4 P08173 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HTT P42858 1/20 0.35
HDAC4 P56524 2/20 0.35
HDAC6 Q9UBN7 1/20 0.35
PPARG P37231 2/20 0.34
PPARD Q03181 1/20 0.34
TSHR P16473 1/20 0.34
GSK3B P49841 1/20 0.34
KDM1A O60341 1/20 0.33
HDAC1 Q13547 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16305096 0.86 PDE2A (0.40) SMN1; SMN2PTGER4PPARAHDAC4HDAC6
SCHEMBL16305069 0.82 PTGER4 (0.52) PTGER4PPARAPPARG
SCHEMBL17684652 0.81 RORC (0.44) PTGER4PPARAPPARG
SCHEMBL16305091 0.80 PTGER4 (0.37) SMN1; SMN2PTGER4PPARACNR1CNR2
SCHEMBL17690477 0.79 NR1H4 (0.48) PTGER4CNR1CNR2PPARG
SCHEMBL17684549 0.75 CCR9 (0.41) PTGER4
SCHEMBL16305088 0.75 RORC (0.48) PTGER4
SCHEMBL17684432 0.74 KDM4E (0.41) SMN1; SMN2PTGER4ALDH1A1
SCHEMBL20113478 0.74 PTGER4 (0.43) PTGER4HDAC6GSK3B
SCHEMBL16305136 0.74 PTGER4 (0.51) PTGER4PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3009426-A1 4-ALKYNYL IMIDAZOLE DERIVATIVE AND MEDICINE COMPRISING SAME AS ACTIVE INGREDIENT Kaken Pharmaceutical Co., Ltd. (JP) 2016-04-20 EP disclosed