SCHEMBL17707484

SCHEMBL17707484

CCCC1(C(O)c2ccc3c(ccn3C(=O)O)c2)CCCN1C(=O)OC(C)(C)C

nearest known ligand 0.33

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 1/20 0.33
GRIN2C Q14957 1/20 0.33
PIK3CD O00329 2/20 0.32
ABL1 P00519 2/20 0.32
EGFR P00533 2/20 0.32
HCK P08631 2/20 0.32
SRC P12931 2/20 0.32
KDR P35968 2/20 0.32
PIK3CA P42336 2/20 0.32
PIK3CB P42338 2/20 0.32
MTOR P42345 2/20 0.32
PIK3CG P48736 2/20 0.32
EPHB4 P54760 2/20 0.32
PRKDC P78527 2/20 0.32
PI4KB Q9UBF8 2/20 0.32
CNR2 P34972 1/20 0.32
NQO1 P15559 1/20 0.30
OXER1 Q8TDS5 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL442590 0.95 PIK3CD (0.36) GRIN2BGRIN2CPIK3CDABL1EGFR
SCHEMBL444534 0.81 SLC6A3 (0.37) GRIN2BGRIN2C
SCHEMBL442630 0.80 GPR119 (0.33) GRIN2BGRIN2CCNR2
SCHEMBL1692041 0.79 CNR2 (0.34) PIK3CDABL1EGFRHCKSRC
SCHEMBL446410 0.78 KCNQ2 (0.39)
SCHEMBL444476 0.76 GRIN2B (0.32) GRIN2BGRIN2CCNR2
SCHEMBL442485 0.76 GRIN2B (0.32) GRIN2BGRIN2CCNR2
SCHEMBL441894 0.75 KCNQ2 (0.36) GRIN2BGRIN2CCNR2
SCHEMBL441389 0.75 GRIN2B (0.32) GRIN2BGRIN2C
SCHEMBL444129 0.75 KCNQ2 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2684871-B1 Heteroaryl pyrrolidinyl and piperidinyl ketone derivatives HOFFMANN LA ROCHE (CH) 2016-05-04 EP disclosed