SCHEMBL17739997

SCHEMBL17739997

O=C(CCOCCOCCOCCOCCn1cc(CN2C(=O)C=CC2=O)nn1)N1CCCC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.40
HRH3 Q9Y5N1 1/20 0.40
CHIT1 Q13231 1/20 0.38
MGLL Q99685 1/20 0.37
DRD2 P14416 5/20 0.36
DRD4 P21917 5/20 0.36
DRD3 P35462 5/20 0.36
HPGD P15428 5/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
ACHE P22303 1/20 0.35
KMT2A Q03164 3/20 0.34
ALDH1A1 P00352 2/20 0.34
RAB9A P51151 2/20 0.34
GAA P10253 1/20 0.34
HSD17B10 Q99714 1/20 0.34
NPC1 O15118 1/20 0.34
LMNA P02545 1/20 0.33
NCF1 P14598 1/20 0.33
TTR P02766 1/20 0.33
IL2 P60568 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19703693 0.89 ALDH1A1 (0.39) HRH4HRH3MGLLDRD2DRD4
SCHEMBL19703576 0.87 TTR (0.36) HRH4HRH3MGLLDRD2DRD4
SCHEMBL19703695 0.86 TTR (0.35) HRH4HRH3CHIT1MGLLDRD2
SCHEMBL19703717 0.85 TTR (0.36) HRH4HRH3DRD2DRD4DRD3
SCHEMBL17739915 0.85 TTR (0.36) HRH4HRH3DRD2DRD4DRD3
SCHEMBL17739959 0.85 TTR (0.36) HRH4HRH3DRD2DRD4DRD3
SCHEMBL19703595 0.84 TTR (0.34) MGLLDRD2DRD4DRD3TTR
SCHEMBL17740210 0.84 TTR (0.36) HRH4HRH3DRD2DRD4DRD3
SCHEMBL17740058 0.83 DRD2 (0.36) HRH4HRH3CHIT1DRD2DRD4
SCHEMBL19703899 0.83 TTR (0.34) HRH4HRH3MGLLDRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016071856-A1 AMATOXIN DERIVATIVES AND CONJUGATES THEREOF AS INHIBITORS OF RNA POLYMERASE NOVARTIS AG (CH) 2016-05-12 WO disclosed