SCHEMBL17744293

SCHEMBL17744293

Nc1cc(Cl)c(OC(F)(F)F)c(Br)c1O

nearest known ligand 0.32

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
WDR5 P61964 1/20 0.32
AKR1C2 P52895 1/20 0.32
AKR1C1 Q04828 1/20 0.32
THRB P10828 1/20 0.31
GAA P10253 1/20 0.31
MMP14 P50281 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13855834 0.80 AKR1C2 (0.32) WDR5AKR1C2AKR1C1
SCHEMBL17744442 0.77 GAA (0.41) THRBGAAMMP14
SCHEMBL17744493 0.77 AKR1C2 (0.32) WDR5AKR1C2AKR1C1THRB
SCHEMBL17744568 0.74 GPR35 (0.43)
SCHEMBL17744451 0.74 GAA (0.34) THRBGAAMMP14
SCHEMBL17744267 0.71 GAA (0.39) THRBGAAMMP14
SCHEMBL29344158 0.70 HSD17B10 (0.37) AKR1C2AKR1C1
SCHEMBL8489664 0.70 AKR1C2 (0.43) WDR5AKR1C2AKR1C1THRBGAA
SCHEMBL24512726 0.70 HSD17B10 (0.44) AKR1C2AKR1C1THRB
SCHEMBL26231908 0.70 WDR5 (0.35) WDR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3020718-B1 NOVEL PDE4 INHIBITOR MEIJI SEIKA PHARMA CO LTD (JP) 2018-12-26 EP disclosed
US-9890142-B2 PDE4 inhibitor MEIJI SEIKA PHARMA CO., LTD. (JP) 2018-02-13 US disclosed
US-9850235-B2 2017-12-26 US disclosed
US-20160159783-A1 PDE4 Inhibitor MEIJI SEIKA PHARMA CO., LTD. (JP) 2016-06-09 US disclosed
EP-3020718-A1 NOVEL PDE4 INHIBITOR Meiji Seika Pharma Co., Ltd. (JP) 2016-05-18 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160159783-A1 PDE4 Inhibitor PDE4A, PDE4B, PDE3B WDR5 2943/4885AKR1C2 627/4885AKR1C1 507/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.