SCHEMBL17748801

SCHEMBL17748801

COc1ccc(/C=C/CCc2ccc(CC(C)C)cc2C)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TUBB1 Q9H4B7 2/20 0.40
ALOX5 P09917 2/20 0.39
PTGS2 P35354 2/20 0.39
PTGS1 P23219 1/20 0.39
KCNH2 Q12809 1/20 0.38
RELA Q04206 2/20 0.38
ESR1 P03372 2/20 0.37
ABL1 P00519 1/20 0.37
TTR P02766 1/20 0.37
CYP1A1 P04798 1/20 0.37
CYP1A2 P05177 1/20 0.37
ABCB1 P08183 1/20 0.37
BCR P11274 1/20 0.37
CYP19A1 P11511 1/20 0.37
NQO2 P16083 1/20 0.37
CYP1B1 Q16678 1/20 0.37
TUBB4A P04350 1/20 0.37
TUBB P07437 1/20 0.37
TUBA3C P0DPH7 1/20 0.37
AHR P35869 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17748803 1.00 TUBB1 (0.40) TUBB1ALOX5PTGS2PTGS1KCNH2
SCHEMBL19491867 0.93 TUBB1 (0.39) TUBB1ALOX5PTGS2PTGS1KCNH2
SCHEMBL9954884 0.83 SLC6A4 (0.46) RELARAB9ASLC6A4LMNATDP1
SCHEMBL9954880 0.83 SLC6A4 (0.46) RELARAB9ASLC6A4LMNATDP1
SCHEMBL23779783 0.78 TLR4 (0.45) AHR
SCHEMBL23779782 0.78 TLR4 (0.45) AHR
SCHEMBL29185869 0.78 SLC6A4 (0.34) SLC6A4
SCHEMBL29185850 0.78 SLC6A4 (0.34) SLC6A4
SCHEMBL9928581 0.75 CYP3A4 (0.57) TUBB1ALOX5PTGS2KCNH2RELA
SCHEMBL7149958 0.73 GABRA1 (0.41) ALOX5PTGS2PTGS1ESR1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3218458-B1 IMPROVMENTS IN OR RELATING TO ORGANIC COMPOUNDS GIVAUDAN SA (CH) 2019-01-02 EP claimed
US-20170298292-A1 IMPROVEMENTS IN OR RELATING TO ORGANIC COMPOUNDS GIVAUDAN S.A. (CH) 2017-10-19 US claimed
EP-3218458-A1 IMPROVMENTS IN OR RELATING TO ORGANIC COMPOUNDS Givaudan S.A. (CH) 2017-09-20 EP claimed
WO-2016074699-A1 IMPROVMENTS IN OR RELATING TO ORGANIC COMPOUNDS GIVAUDAN SA (CH) 2016-05-19 WO claimed
EP-3218458-B1 IMPROVMENTS IN OR RELATING TO ORGANIC COMPOUNDS GIVAUDAN SA (CH) 2019-01-02 EP disclosed
EP-3218458-B1 IMPROVMENTS IN OR RELATING TO ORGANIC COMPOUNDS GIVAUDAN SA (CH) 2019-01-02 EP disclosed
US-10119097-B2 Organic compounds GIVAUDAN S.A. (CH) 2018-11-06 US disclosed
US-20170298292-A1 IMPROVEMENTS IN OR RELATING TO ORGANIC COMPOUNDS GIVAUDAN S.A. (CH) 2017-10-19 US disclosed
US-20170298292-A1 IMPROVEMENTS IN OR RELATING TO ORGANIC COMPOUNDS GIVAUDAN S.A. (CH) 2017-10-19 US disclosed
US-20170298292-A1 IMPROVEMENTS IN OR RELATING TO ORGANIC COMPOUNDS GIVAUDAN S.A. (CH) 2017-10-19 US disclosed
EP-3218458-A1 IMPROVMENTS IN OR RELATING TO ORGANIC COMPOUNDS Givaudan S.A. (CH) 2017-09-20 EP disclosed
WO-2016074699-A1 IMPROVMENTS IN OR RELATING TO ORGANIC COMPOUNDS GIVAUDAN SA (CH) 2016-05-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10119097-B2 Organic compounds OR10J3, CBR3, C9 TUBB1 1029/4885ALOX5 228/4885PTGS2 1229/4885
US-20170298292-A1 IMPROVEMENTS IN OR RELATING TO ORGANIC COMPOUNDS OR10J3, C5, CBR3 TUBB1 784/4885ALOX5 224/4885PTGS2 1091/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.