SCHEMBL17749545

SCHEMBL17749545

N=c1n(CCN2CCCCC2)c2ccccc2n1CC(O)COc1ccc(Cl)cc1Cl

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 9/20 1.00
TP53 P04637 8/20 1.00
MAPT P10636 4/20 1.00
F8 P00451 1/20 1.00
F5 P12259 1/20 1.00
TSHR P16473 7/20 0.69
LMNA P02545 4/20 0.68
MEN1 O00255 4/20 0.68
KMT2A Q03164 4/20 0.68
NPSR1 Q6W5P4 4/20 0.68
GAA P10253 1/20 0.68
IDE P14735 1/20 0.68
XBP1 P17861 1/20 0.68
PAX8 Q06710 1/20 0.68
ALOX15 P16050 1/20 0.67
CYP1A2 P05177 1/20 0.63
CYP2D6 P10635 1/20 0.63
ALDH1A1 P00352 2/20 0.63
HTT P42858 1/20 0.57
MITF O75030 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2568428 0.86 SMN1; SMN2 (0.84) SMN1; SMN2TP53MAPTF8F5
SCHEMBL7629030 0.85 SMN1; SMN2 (0.82) SMN1; SMN2TP53MAPTF8F5
SCHEMBL17749503 0.85 SMN1; SMN2 (0.74) SMN1; SMN2TP53MAPTF8F5
SCHEMBL17749595 0.83 SMN1; SMN2 (0.70) SMN1; SMN2TP53MAPTF8F5
SCHEMBL2505043 0.82 LMNA (0.98) SMN1; SMN2TP53MAPTF8F5
SCHEMBL17761713 0.81 TP53 (0.71) SMN1; SMN2TP53MAPTF8F5
SCHEMBL17749565 0.81 TP53 (0.71) SMN1; SMN2TP53MAPTF8F5
SCHEMBL17761742 0.81 TP53 (0.71) SMN1; SMN2TP53MAPTF8F5
SCHEMBL17749492 0.80 LMNA (0.73) SMN1; SMN2TP53MAPTF8F5
SCHEMBL17761945 0.80 SMN1; SMN2 (0.66) SMN1; SMN2TP53MAPTF8F5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016077541-A1 NOVEL ANTI-INFECTIVE COMPOUNDS AND METHODS USING SAME THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2016-05-19 WO claimed
WO-2016077541-A1 NOVEL ANTI-INFECTIVE COMPOUNDS AND METHODS USING SAME THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2016-05-19 WO disclosed
WO-2016077541-A1 NOVEL ANTI-INFECTIVE COMPOUNDS AND METHODS USING SAME THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2016-05-19 WO disclosed