SCHEMBL1775654

SCHEMBL1775654

COc1ccc(S(=O)(=O)Nc2ccc(OC3CCCNC3)c3ccccc23)cc1

nearest known ligand 0.59

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 16/20 0.59
NFE2L2 Q16236 9/20 0.59
SQSTM1 Q13501 2/20 0.59
GAA P10253 2/20 0.53
MITF O75030 1/20 0.53
ALDH1A1 P00352 1/20 0.53
LMNA P02545 1/20 0.53
TP53 P04637 1/20 0.53
MAPT P10636 1/20 0.53
THRB P10828 1/20 0.53
HPGD P15428 1/20 0.53
ALOX15 P16050 1/20 0.53
CASP1 P29466 1/20 0.53
GFER P55789 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
HKDC1 Q2TB90 1/20 0.53
HSD17B10 Q99714 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.53
HTR6 P50406 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL1776067 0.99 KEAP1 (0.58) KEAP1NFE2L2SQSTM1GAAMITF
SCHEMBL1775785 0.94 KEAP1 (0.61) KEAP1NFE2L2SQSTM1GAAMITF
Hydrochloric Acid SCHEMBL1773873 0.93 KEAP1 (0.60) KEAP1NFE2L2SQSTM1GAAMITF
SCHEMBL1775005 0.88 HKDC1 (0.49) KEAP1NFE2L2SQSTM1ALDH1A1LMNA
Hydrochloric Acid SCHEMBL1776019 0.87 HKDC1 (0.48) KEAP1NFE2L2SQSTM1ALDH1A1LMNA
SCHEMBL1777498 0.82 HKDC1 (0.51) KEAP1NFE2L2SQSTM1ALDH1A1HKDC1
SCHEMBL1774701 0.82 HKDC1 (0.51) KEAP1NFE2L2SQSTM1ALDH1A1HKDC1
SCHEMBL1776585 0.82 HKDC1 (0.51) KEAP1NFE2L2SQSTM1ALDH1A1HKDC1
Hydrochloric Acid SCHEMBL1775345 0.81 HKDC1 (0.50) KEAP1NFE2L2SQSTM1HKDC1
Hydrochloric Acid SCHEMBL1775351 0.81 HKDC1 (0.50) KEAP1NFE2L2SQSTM1HKDC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7943639-B2 Such as 6-benzenesulfonyl-4-piperazin-1-yl-quinoline hydrochloride; for treatment of central nervous system and/or 5- HT6 receptor related disorders; for weight gain/loss PROXIMAGEN LIMITED (GB) 2011-05-17 US claimed